Affinity DataKi: 0.120nMAssay Description:Mixed-type inhibition of bovine xanthine oxidaseMore data for this Ligand-Target Pair
TargetEcdysone receptor/Protein ultraspiracle homolog(Choristoneura fumiferana)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Binding affinity to Choristoneura fumiferana EcRMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Mixed-type inhibition of bovine xanthine oxidase assessed as enzyme-inhibitor complexMore data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Chilo suppressalis)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Chilo suppressalis (rice stem borer) EcRMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine milk xanthine oxidoreductase by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity towards mu opioid receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetEcdysone receptor/USP(Plodia interpunctella)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Plodia interpunctella (Indian meal moth ) EcRMore data for this Ligand-Target Pair
TargetEcdysone receptor/Gene regulation protein(Heliothis virescens)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Heliothis virescens (tobacco budworm) EcRMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Competitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using varying levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetEcdysone receptor/Ultraspiracle(Chironomus tentans)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to Chironomus tentans EcRMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
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