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Found 3393 with Last Name = 'hill' and Initial = 'r'
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University of California

Curated by ChEMBL
LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  0.120nMAssay Description:Mixed-type inhibition of bovine xanthine oxidaseMore data for this Ligand-Target Pair
TargetEcdysone receptor/Protein ultraspiracle homolog(Choristoneura fumiferana)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  0.501nMAssay Description:Binding affinity to Choristoneura fumiferana EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University of California

Curated by ChEMBL
LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  0.900nMAssay Description:Mixed-type inhibition of bovine xanthine oxidase assessed as enzyme-inhibitor complexMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50006730((R)-2-Hydroxymethyl-5-[6-(1-methyl-2-phenyl-ethyla...)
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
In DepthDetails PubMed
TargetEcdysone receptor/Ultraspiracle(Chilo suppressalis)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Chilo suppressalis (rice stem borer) EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122928(5-{6-[5-Chloro-2-(3-methyl-isoxazol-5-ylmethoxy)-b...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University of California

Curated by ChEMBL
LigandPNGBDBM50497925(CHEBI:70981 | CHEMBL3314206)
Affinity DataKi:  1.80nMAssay Description:Inhibition of bovine milk xanthine oxidoreductase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards mu opioid receptor was determinedMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50034171(3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182312((2S,3S,4R,5R)-5-(6-(3,5-dichlorobenzylamino)-9H-pu...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018786(CHEMBL538309 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/USP(Plodia interpunctella)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Plodia interpunctella (Indian meal moth ) EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Gene regulation protein(Heliothis virescens)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Heliothis virescens (tobacco budworm) EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182322((2S,3S,4R,5R)-5-(6-(2,5-dimethoxybenzylamino)-9H-p...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82557(I-ABA | IABA | N(6)-(4-Amino-3-iodobenzyl)adenosin...)
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018768(CHEMBL556957 | N-(2-Azepan-1-yl-cyclohexyl)-2-(4-c...)
Affinity DataKi:  4nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122927((2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methyla...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122927((2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methyla...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82557(I-ABA | IABA | N(6)-(4-Amino-3-iodobenzyl)adenosin...)
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018767(CHEMBL535581 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122926(3-Amino-5-{6-[5-chloro-2-(3-methyl-isoxazol-5-ylme...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50037785(2-(6-{[2-(4-aminophenyl)ethyl]amino}-9H-purin-9-yl...)
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018771(CHEMBL535801 | N-(2-Azepan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182326((2S,3S,4R,5R)-5-(6-(2-(2-amino-2-oxoethoxy)-5-chlo...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017495(2-Benzo[b]thiophen-4-yl-N-[2-(3-hydroxymethyl-pyrr...)
Affinity DataKi:  7nMAssay Description:Binding affinity towards opioid receptor kappa was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50180955(CHEMBL3818617)
Affinity DataKi:  8nMAssay Description:Competitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using varying levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182313((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-(4-(dimethylamin...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182324((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-oxo-2-(piperazin...)
Affinity DataKi:  9.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle(Chironomus tentans)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  10nMAssay Description:Binding affinity to Chironomus tentans EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018781(CHEMBL557426 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  12nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50017500(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  14nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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