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Found 84 with Last Name = 'amemiya' and Initial = 'y'
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50001922(2-Naphthalen-1-ylmethyl-4,5-dihydro-1H-imidazole; ...)
Affinity DataIC50:  0.00110nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230389(CHEMBL541105)
Affinity DataIC50:  0.00340nMAssay Description:Compound was tested for Adrenergic activity against Alpha-2 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230393(CHEMBL553231)
Affinity DataIC50:  0.0140nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230395(CHEMBL557985)
Affinity DataIC50:  0.0160nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230388(CHEMBL537830)
Affinity DataIC50:  0.0340nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230394(CHEMBL538801)
Affinity DataIC50:  0.120nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230392(CHEMBL554581)
Affinity DataIC50:  0.260nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50230391(CHEMBL164540)
Affinity DataIC50:  0.610nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049128(5-(1-Hydroxy-ethyl)-2-propyl-3-[2'-(2H-tetrazol-5-...)
Affinity DataIC50:  4.90nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049118(2-Ethyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...)
Affinity DataIC50:  5.30nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018179(2-Imidazol-1-ylmethyl-4,5-dihydro-benzo[b]thiophen...)
Affinity DataIC50:  6nMAssay Description:Inhibition of platelet microsomal thromboxane A synthetase in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049123(5-Hydroxymethyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-...)
Affinity DataIC50:  6.90nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50241364(4-(1-hydroxy-1-methylethyl)-2-propyl-1-{[2'-(1H-te...)
Affinity DataIC50:  8.10nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049107(2-Propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  9.10nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049109(2-Butyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...)
Affinity DataIC50:  9.5nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049124(5-Methyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  11nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049116(5-Ethyl-2-propyl-3-(2'-tetrazol-1-yl-biphenyl-4-yl...)
Affinity DataIC50:  12nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018179(2-Imidazol-1-ylmethyl-4,5-dihydro-benzo[b]thiophen...)
Affinity DataIC50:  13nMAssay Description:Inhibition of platelet microsomal thromboxane A2 synthetase in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018179(2-Imidazol-1-ylmethyl-4,5-dihydro-benzo[b]thiophen...)
Affinity DataIC50:  13nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018181(2-Imidazol-1-ylmethyl-4,5,6,7-tetrahydro-benzo[b]t...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet microsomal thromboxane A synthetase in humansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  22nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018181(2-Imidazol-1-ylmethyl-4,5,6,7-tetrahydro-benzo[b]t...)
Affinity DataIC50:  26nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018181(2-Imidazol-1-ylmethyl-4,5,6,7-tetrahydro-benzo[b]t...)
Affinity DataIC50:  26nMAssay Description:Inhibition of platelet microsomal thromboxane A synthetase in humansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049112(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-et...)
Affinity DataIC50:  28nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049132(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-1-...)
Affinity DataIC50:  28nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049122(2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-(1-hy...)
Affinity DataIC50:  30nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049117(3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-ethyl-5-(1-hy...)
Affinity DataIC50:  37nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049130(5-Isopropyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  46nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049113(5-Isopropenyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-bi...)
Affinity DataIC50:  50nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049106(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-1-...)
Affinity DataIC50:  51nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049108(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl...)
Affinity DataIC50:  58nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049108(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-hydroxymethyl...)
Affinity DataIC50:  58nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049126(3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-propyl-3H-imi...)
Affinity DataIC50:  60nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50282291(2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-hydro...)
Affinity DataIC50:  65nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018183(2-Imidazol-1-ylmethyl-4,5,6,7-tetrahydro-benzo[b]t...)
Affinity DataIC50:  86nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018186(2-Imidazol-1-ylmethyl-6,7-dihydro-benzo[b]thiophen...)
Affinity DataIC50:  93nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049110(2-Propyl-1-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  100nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049103(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-ethyl-2-propy...)
Affinity DataIC50:  100nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018178(2-(2-Imidazol-1-yl-ethyl)-6,7-dihydro-benzo[b]thio...)
Affinity DataIC50:  100nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM7962(4-(2-Imidazol-1-yl-ethoxy)-benzoic acid; hydrochlo...)
Affinity DataIC50:  106nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM7962(4-(2-Imidazol-1-yl-ethoxy)-benzoic acid; hydrochlo...)
Affinity DataIC50:  106nMAssay Description:Inhibition of platelet microsomal thromboxane A2 synthetase in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049129(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-ethyl-1-hy...)
Affinity DataIC50:  110nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049104(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-methyl-2-prop...)
Affinity DataIC50:  110nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018176(2-(Imidazol-1-yl-phenyl-methyl)-6,7-dihydro-benzo[...)
Affinity DataIC50:  114nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50018184(5-Imidazol-1-ylmethyl-4,5,6,7-tetrahydro-benzo[b]t...)
Affinity DataIC50:  114nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  120nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50009505(2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-chlor...)
Affinity DataIC50:  130nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50009505(2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-chlor...)
Affinity DataIC50:  130nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
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