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Found 23 with Last Name = 'arvedson' and Initial = 's'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146490(3-(S)-Benzo[1,3]dioxol-5-yl-3-({(R)-5-oxo-1-[3-(1,...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146492(3-Benzo[1,3]dioxol-5-yl-3-({1-[2-fluoro-5-(1,4,5,6...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146497(3-Benzo[1,3]dioxol-5-yl-3-({5-oxo-1-[3-(1,4,5,6-te...)
Affinity DataKi:  0.700nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146493(3-({5-Oxo-1-[3-(1,4,5,6-tetrahydro-pyrimidin-2-yla...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146481(3-Benzo[1,3]dioxol-5-yl-3-({1-[3-(3-benzyl-ureido)...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146488(3-{[1-(2-Fluoro-5-guanidino-phenyl)-5-oxo-pyrrolid...)
Affinity DataKi:  2.90nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146482(3-({1-[3-(4,5-Dihydro-1H-imidazol-2-ylamino)-pheny...)
Affinity DataKi:  5.10nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146485(3-(R)-Benzo[1,3]dioxol-5-yl-3-({(R)-5-oxo-1-[3-(1,...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146496((S)-3-({(R)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi:  10nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146495(3-({1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-pyrrolidi...)
Affinity DataKi:  10nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146484(3-({1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-pyrrolidi...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146489(3-{[1-(3-Guanidino-phenyl)-5-oxo-pyrrolidine-3-car...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146494(3-{[1-(2-Chloro-5-guanidino-phenyl)-5-oxo-pyrrolid...)
Affinity DataKi:  53nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146491(3-({1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-pyrrolidi...)
Affinity DataKi:  71nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146483((R)-3-({(R)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi:  154nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146486((S)-3-({(S)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146487(3-({(S)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-pyrro...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146490(3-(S)-Benzo[1,3]dioxol-5-yl-3-({(R)-5-oxo-1-[3-(1,...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146486((S)-3-({(S)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146496((S)-3-({(R)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146487(3-({(S)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-pyrro...)
Affinity DataKi: >2.50E+4nMAssay Description:Affinity for alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146485(3-(R)-Benzo[1,3]dioxol-5-yl-3-({(R)-5-oxo-1-[3-(1,...)
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50146483((R)-3-({(R)-1-[3-(3-Benzyl-ureido)-phenyl]-5-oxo-p...)
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity towards vitronectin receptor (AlphaV-beta3 integrin).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed