Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of hypoxia induced HIF1 transcriptional activity in human Hep3B cells by cell-based HRE reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 829nMAssay Description:Inhibition of human chymaseMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human chymaseMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of hypoxia induced HIF1 transcriptional activity in human Hep3B cells by cell-based HRE reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory concentration against human PTP1B expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.82E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory concentration against human PTP1B expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Rattus norvegicus (rat))
Dongguk University-Seoul
Curated by ChEMBL
Dongguk University-Seoul
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of DGAT in rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory concentration against human PTP1B expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.21E+3nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human macrophage ACAT expressed in human HepG2 cells using [14C]oleoyl-CoA as substrate incubated for 20 mins prior to substrate additi...More data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Molecular Cancer Research Center
Curated by ChEMBL
Molecular Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of hypoxia induced HIF1alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair