Affinity DataKi: 3.20nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 20nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 25nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 43nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 59nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 78nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 92nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 100nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 110nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 110nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 130nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 140nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 150nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 210nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 220nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 230nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 260nMpH: 5.0Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 5 after 1.5 hrs by Microbeta liquid scintillation counting...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 300nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 340nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 360nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 370nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 390nMpH: 6.4Assay Description:Displacement of [3H]BMS-599240 from BACE1 (unknown origin) expressed in HEK293 cells at pH 6.4 after 1.5 hrs by Microbeta liquid scintillation counti...More data for this Ligand-Target Pair