Affinity DataKi: 1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 990nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 4 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 4 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 5 receptor expressed in HEK293 cells; N = 4More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 1 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 3 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 5 receptor expressed in HEK293 cells; N = 4More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 5 receptor expressed in HEK293 cells; N = 4More data for this Ligand-Target Pair