Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 6.31E+3nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Activity at vasopressin V1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Activity at vasopressin V1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 4.50E+3nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 8.00E+3nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair
Affinity DataKd: 5.50E+3nMAssay Description:Binding affinity towards FK506 binding protein 12 as measured by displacement of a radiolabelled FK506 analogueMore data for this Ligand-Target Pair