Affinity DataKi: 82nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Inhibition of peroxidase activity of MPO isolated from human polynuclear leukocytes using Amplex Red as substrate assessed as formation of resorufin ...More data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin...More data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Concentration required for 50% in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Concentration required for 50% in vitro activity against rat SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of KHK (unknown origin) using D-fructose as substrate after 60 mins in presence of ATP by LC-MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Concentration required for 50% for in vitro activity against human SDH (sorbitol dehydrogenase)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GPR40 expressed HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair