Affinity DataKi: 32nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 200nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAdenosine receptor A1(BOVINE)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 501nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Affinity DataKi: 794nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAdenosine receptor A1(BOVINE)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M1(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M1(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(PIG)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetVoltage-dependent calcium channel gamma-1 subunit(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetVoltage-dependent calcium channel gamma-1 subunit(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetVoltage-dependent calcium channel gamma-1 subunit(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(RAT)
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database
Center For Bio-Pharmaceutical Sciences
Curated by PDSP Ki Database