Affinity DataKi: 0.200nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [131I]-(R)-8More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [3H]SR-141,716AMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [131I]-(R)-8More data for this Ligand-Target Pair
Affinity DataKi: 1.91nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of N-terminal His tagged human Pin1 expressed in Escherichia coli BL21 (DE3) using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate preincu...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA as substrate preincubated with enzyme for 12 hrs followed by substrate ...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [3H]SR-141,716AMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA as substrate preincubated with enzyme for 12 hrs followed by substrate ...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of Escherichia coli PDFMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 820nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA, Suc-Ala-Glu-Pro-Phe-pNA or Suc-Ala-Ala-Pro-Phe-pNA as substrate preinc...More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: 9.60E+3nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human PARP-1 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human PARP-1 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair