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Found 8 with Last Name = 'daniel' and Initial = 'bj'
TargetMitogen-activated protein kinase(Toxoplasma gondii)
Tulane University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Toxoplasma gondii recombinant MAPK1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase(Toxoplasma gondii)
Tulane University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50295553(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Toxoplasma gondii recombinant MAPK1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Tulane University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM13531(4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridy...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant p38alpha assessed as [gamma33P]ATP utilization by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Tulane University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50295553(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant p38alpha assessed as [gamma33P]ATP utilization by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50519517(CHEMBL4461111)
Affinity DataIC50:  4.87E+3nMAssay Description:Inhibition of cathepsin B (unknown origin) assessed as reduction in enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Tulane University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human recombinant p38alpha assessed as [gamma33P]ATP utilization by microplate scintillation countingMore data for this Ligand-Target Pair
TargetSortase family protein(Staphylococcus aureus)
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50519515(CHEMBL4474465)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus ATCC 6538p sortase A incubated for 1 hr in presence of (Dabcyl-QALPETGEE-Edans substrate by fluoresce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50519516(CHEMBL4434939)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus ATCC 6538p sortase A incubated for 1 hr in presence of (Dabcyl-QALPETGEE-Edans substrate by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed