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Found 100 with Last Name = 'darwish' and Initial = 'ss'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237049(CHEMBL3133904)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237048(CHEMBL3132872)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469211(CHEMBL4283503)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237123(CHEMBL4097369)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237111(CHEMBL4103464)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237097(CHEMBL4075530)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237186(CHEMBL4092951)
Affinity DataIC50:  9.10nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237098(CHEMBL4075103)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237108(CHEMBL4065288)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237124(CHEMBL4091921)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50179494(CHEMBL3815163)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466167(CHEMBL4278808)
Affinity DataIC50:  12nMAssay Description:Inhibition of Haspin (unknown origin) after 3 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466158(CHEMBL4290247)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466158(CHEMBL4290247)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human Dyrk1A expressed in Baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466158(CHEMBL4290247)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466168(CHEMBL4282366)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237062(CHEMBL4076434)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237063(CHEMBL4102455)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237047(CHEMBL4088718)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration against rabbit muscle glyceraldehyde-3-phosphate dehydrogenase (GAPDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM138364(US10278929, Compound 12 | US11337935, Compound 12 ...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant full length His-tagged PIM-1 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469213(CHEMBL4278353)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237112(CHEMBL4089588)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237096(CHEMBL4097862)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237117(CHEMBL4078182)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using KHKKLAEGSA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237121(CHEMBL4101774)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466164(CHEMBL4283474)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237099(CHEMBL4066504)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237110(CHEMBL4062528)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237109(CHEMBL4071170)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469215(CHEMBL4281810)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237188(CHEMBL4088760)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using KHKKLAEGSA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466158(CHEMBL4290247)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human Haspin expressed in Baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237052(CHEMBL4072769)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466157(CHEMBL4294049)
Affinity DataIC50:  37nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237117(CHEMBL4078182)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469211(CHEMBL4283503)
Affinity DataIC50:  43nMAssay Description:Inhibition of DYRK1A in human HeLa cells harboring GFP-SF3b1-NT assessed as reduction in SF3b1 phosphorylation at T343 residue after 18 hrs by Wester...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469218(CHEMBL4287985)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469214(CHEMBL4292442)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466169(CHEMBL4295177)
Affinity DataIC50:  49nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237105(CHEMBL4067514)
Affinity DataIC50:  49nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50466159(CHEMBL4292471)
Affinity DataIC50:  51nMAssay Description:Inhibition of recombinant full length human Dyrk1A expressed in Baculovirus expression system using KKISGRLSPIMTEQ as substrate in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237113(CHEMBL4092966)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469217(CHEMBL4294080)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21(DE3) using KKISGRLSPIMTEQ-NH2 as substrate after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237187(CHEMBL4065300)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using KHKKLAEGSA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237102(CHEMBL4085352)
Affinity DataIC50:  61nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50237058(CHEMBL4080711)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant GST-tagged EGFR (668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469214(CHEMBL4292442)
Affinity DataIC50:  67nMAssay Description:Inhibition of full length recombinant human GST-tagged DYRK1B expressed in baculovirus expression system using KKISGRLSPIMTEQ-NH2 as substrate after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469211(CHEMBL4283503)
Affinity DataIC50:  73nMAssay Description:Inhibition of full length recombinant human GST-tagged DYRK1B expressed in baculovirus expression system using KKISGRLSPIMTEQ-NH2 as substrate after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469211(CHEMBL4283503)
Affinity DataIC50:  76nMAssay Description:Inhibition of human GST-tagged haspin expressed in baculovirus expression system in presence of 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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