Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMpH: 7.4Assay Description:Inhibitory activity against human plasma renin at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMpH: 7.4Assay Description:Inhibitory activity against human plasma renin at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMpH: 6.5Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMpH: 6.0Assay Description:Inhibitory activity against purified human renal renin at pH 6.0More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMpH: 6.0Assay Description:Inhibitory activity against purified human plasma renin at pH 6.0More data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMpH: 6.5Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMpH: 6.0Assay Description:Inhibitory activity against purified human plasma renin at pH 6.0More data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMpH: 6.0Assay Description:Inhibitory activity against purified human plasma renin at pH 6.0More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMpH: 7.4Assay Description:Inhibitory activity against human plasma renin at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMpH: 6.5Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMpH: 6.5Assay Description:Compound was evaluated for the inhibitory concentration against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMpH: 6.0Assay Description:Inhibitory activity against purified human plasma renin at pH 6.0More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMpH: 6.5Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMpH: 6.0Assay Description:In vitro potency against plasma renin at a pH of 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMpH: 6.0Assay Description:In vitro activity against human renin (pH 6.0)More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMpH: 7.4Assay Description:In vitro potency against purified renin at a pH of 6.0.More data for this Ligand-Target Pair
Affinity DataIC50: 0.990nMpH: 6.5Assay Description:Compound was evaluated for the inhibitory concentration against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 0.990nMpH: 6.5Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.0Assay Description:In vitro activity against human renin (pH 6.0)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.0Assay Description:In vitro potency against plasma renin at a pH of 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.0Assay Description:In vitro potency against human plasma renin at a pH of 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 6.0Assay Description:In vitro potency against human plasma renin at a pH of 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Abbvie Bioresearch Center
Curated by ChEMBL
Abbvie Bioresearch Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-fused human recombinant ROCK2 (11 to 552 residues) expressed in Spodoptera frugiperda insect cells using STK S2 peptide substrate a...More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Abbvie Bioresearch Center
Curated by ChEMBL
Abbvie Bioresearch Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of ROCK1 (unknown origin) incubated for 2 hrs by AbbVie kinase panel assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Abbvie Bioresearch Center
Curated by ChEMBL
Abbvie Bioresearch Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-fused human recombinant ROCK2 (11 to 552 residues) expressed in Spodoptera frugiperda insect cells using STK S2 peptide substrate a...More data for this Ligand-Target Pair
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Abbvie Bioresearch Center
Curated by ChEMBL
Abbvie Bioresearch Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of ROCK2 (unknown origin) incubated for 2 hrs by AbbVie kinase panel assayMore data for this Ligand-Target Pair
TargetcGMP-dependent protein kinase 1(Homo sapiens (Human))
Abbvie Bioresearch Center
Curated by ChEMBL
Abbvie Bioresearch Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PKG1A (unknown origin) incubated for 2 hrs by AbbVie kinase panel assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against human renal renin using radioimmuno assay for angiotensin I productionMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMpH: 6.0Assay Description:In vitro activity against human renin (pH 6.0)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMpH: 7.4Assay Description:Inhibitory activity against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMpH: 6.5Assay Description:Compound was evaluated for the inhibitory concentration against purified human renal renin at pH 6.5More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMpH: 6.0Assay Description:In vitro potency against purified renin at a pH of 7.4More data for this Ligand-Target Pair