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Found 70 with Last Name = 'emal' and Initial = 'cd'
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  4.10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  6.60nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  7nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  8nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50:  10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50:  10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50:  12nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  14nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  18nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50:  20nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50:  28nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92482(CDE-008 | US9120744, CDE-008)
Affinity DataIC50:  44nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50:  74nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  79nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50:  86nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  91nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50:  116nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50:  132nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92482(CDE-008 | US9120744, CDE-008)
Affinity DataIC50:  162nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50:  174nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310309(CHEMBL596879 | N-(3,4-dihydroxyphenylsulfonyl)-N-h...)
Affinity DataIC50:  284nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92480(Epigallocatechin-3,5-Digallate, C)
Affinity DataIC50:  330nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310311(CHEMBL601265 | N-cyclohexyl-N-(3,4-dihydroxyphenyl...)
Affinity DataIC50:  594nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50:  644nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University of Michigan

LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50:  758nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310308(CHEMBL597478 | N-(3,4-dihydroxyphenylsulfonyl)-3,4...)
Affinity DataIC50:  2.67E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM31712(HEXACHLOROPHENE | Hexach-lorophene | MLS000028433 ...)
Affinity DataIC50:  3.80E+3nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50041419(1,2,5,8-tetrahydroxy-9,10-anthracenedione | 1,2,5,...)
Affinity DataIC50:  4.40E+3nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310310(CHEMBL596880 | N-benzyl-N-(3,4-dihydroxyphenylsulf...)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50085536(3,4,5-Trihydroxybenzoate, X | 3,4,5-trihydroxybenz...)
Affinity DataIC50:  6.60E+3nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310301(CHEMBL599742 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50:  9.32E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92482(CDE-008 | US9120744, CDE-008)
Affinity DataIC50: >1.00E+4nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50: >1.00E+4nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  1.18E+4nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  1.54E+4nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92481(Sennoside A, G)
Affinity DataIC50:  5.10E+4nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310307(CHEMBL596861 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50: >3.00E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50: >3.00E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50: >3.00E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310299(CHEMBL599342 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310305(CHEMBL596859 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-4...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
University of Michigan

LigandPNGBDBM50310306(CHEMBL611972 | N,N'-(ethane-1,2-diyl)bis(N-ethylbe...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310299(CHEMBL599342 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-3...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310312(CHEMBL597509 | N,N'-bis(3,4-dihydroxybenzenesulfon...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310305(CHEMBL596859 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-4...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310313(CHEMBL596860 | N,N'-(ethane-1,2-diyl)bis(N-ethyl-2...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310306(CHEMBL611972 | N,N'-(ethane-1,2-diyl)bis(N-ethylbe...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310310(CHEMBL596880 | N-benzyl-N-(3,4-dihydroxyphenylsulf...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAntithrombin-III(Homo sapiens (Human))
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310311(CHEMBL601265 | N-cyclohexyl-N-(3,4-dihydroxyphenyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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