Affinity DataKi: 0.0460nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0585nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0637nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.122nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.127nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.131nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.143nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.183nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.198nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.280nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Inhibition of Protein kinase C alpha expressed in Sf-9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.367nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nM ΔG°: -53.8kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Agonist activity at human CB2 receptor transfected in CHO cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 min...More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Inhibition of FITC-labeled BH3 peptide binding to human MCL1 expressed in Escherichia coli BL21 (DE3) incubated for 0.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human Bcl-xl expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins follow...More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human Bcl-2 expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins followe...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human MCL1 expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins followed...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKi: <1.20nMAssay Description:Binding affinity to full length human MCL1 (173 to 321 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant incubated f...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh
Curated by PDSP Ki Database
University of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Agonist activity at CB1 receptor in mouse Neuro2a cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 mins by liq...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 1.85nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair