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Found 1113 with Last Name = 'fan' and Initial = 'w'
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485941(CHEMBL2181004)
Affinity DataKi:  0.0460nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485945(CHEMBL2181003)
Affinity DataKi:  0.0585nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485942(CHEMBL2181002)
Affinity DataKi:  0.0637nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485950(CHEMBL2181009)
Affinity DataKi:  0.122nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485944(CHEMBL2181006)
Affinity DataKi:  0.127nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485943(CHEMBL2181001)
Affinity DataKi:  0.131nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485946(CHEMBL2181000)
Affinity DataKi:  0.143nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485947(CHEMBL2181008)
Affinity DataKi:  0.183nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485949(CHEMBL2180999)
Affinity DataKi:  0.198nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485948(CHEMBL2181007)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Wuhan University Of Technology

Curated by ChEMBL
LigandPNGBDBM50537515(CHEMBL4644088)
Affinity DataKi:  0.300nMAssay Description:Inhibition of Protein kinase C alpha expressed in Sf-9 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485940(CHEMBL2181005)
Affinity DataKi:  0.367nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239073(US9416103, CP-55,940)
Affinity DataKi:  0.370nM ΔG°:  -53.8kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.470nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.470nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  0.610nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50036649((7R,10S)-1-(6-fluorobenzo[d]isoxazol-3-yl)-4-[5-fl...)
Affinity DataKi:  0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50036649((7R,10S)-1-(6-fluorobenzo[d]isoxazol-3-yl)-4-[5-fl...)
Affinity DataKi:  0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50036648((7R,10S)-4-[5-fluoro-9,15-diazatetracyclo[10.2.1.0...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  0.810nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  0.810nMAssay Description:Agonist activity at human CB2 receptor transfected in CHO cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50046475(4-[9,15-diazatetracyclo[10.2.1.02,10.03,8]pentadec...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50297345((5S,8S,13R,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50047457(4-[9,16-diazatetracyclo[10.3.1.02,10.03,8]hexadeca...)
Affinity DataKi:  0.850nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50244168(CHEMBL4073496 | US10533010, Example I-239 | US1120...)
Affinity DataKi: <1nMAssay Description:Inhibition of FITC-labeled BH3 peptide binding to human MCL1 expressed in Escherichia coli BL21 (DE3) incubated for 0.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human Bcl-xl expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human Bcl-2 expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50078163(CHEMBL3417704)
Affinity DataKi: <1nMAssay Description:Binding affinity to full length human MCL1 expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant preincubated for 30 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50581350(CHEMBL5079948)
Affinity DataKi: <1.20nMAssay Description:Binding affinity to full length human MCL1 (173 to 321 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50047436(8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-8-aza-bicyclo[...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  1.70nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50036647((7R,10S)-5-[9,15-diazatetracyclo[10.2.1.02,10.03,8...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  1.70nMAssay Description:Agonist activity at CB1 receptor in mouse Neuro2a cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 mins by liq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50036648((7R,10S)-4-[5-fluoro-9,15-diazatetracyclo[10.2.1.0...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(CHEMBL216640 | Dyn A(1-11)-NH2 | Dynorphin A analo...)
Affinity DataKi:  1.85nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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