Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair