TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.87nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by ChEMBL
Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 13.5nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair