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Found 908 with Last Name = 'favata' and Initial = 'm'
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269976(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Ly...)
Affinity DataIC50:  6.87nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141397(4-({3-[(Z)-2-Amino-2-(2-amino-phenylsulfanyl)-1-cy...)
Affinity DataIC50:  7nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269975(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Ly...)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141438(4-({3-[(Z)-2-Amino-1-cyano-2-(2-hydroxy-phenylsulf...)
Affinity DataIC50:  8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141412((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-{3-[hydro...)
Affinity DataIC50:  8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141406((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-{3-[(2,4-...)
Affinity DataIC50:  8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141410((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  12nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141441(3-({3-[(Z)-2-Amino-2-(2-amino-phenylsulfanyl)-1-cy...)
Affinity DataIC50:  13nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269978(Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fl...)
Affinity DataIC50:  13.5nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141404(4-({3-[(Z)-2-Amino-2-(2-amino-phenylsulfanyl)-1-cy...)
Affinity DataIC50:  14nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141426((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141400((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-{3-[hydro...)
Affinity DataIC50:  17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141417((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141440((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  24nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141399((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-{3-[(2,3-...)
Affinity DataIC50:  25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141427((Z)-3-Amino-2-{3-[hydroxy-(3-nitro-phenyl)-methyl]...)
Affinity DataIC50:  25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141401((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141418((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  30nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141431((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-(3-{hydro...)
Affinity DataIC50:  35nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141419((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-(3-phenox...)
Affinity DataIC50:  40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141437((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-(3-benzyl...)
Affinity DataIC50:  40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141416((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-{3-[(3-fl...)
Affinity DataIC50:  44nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141425((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  47nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute

Curated by ChEMBL
LigandPNGBDBM50141415((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)
Affinity DataIC50:  50nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576872(4-(1-(2-Chloro-4-((((1- ethyl-1H-pyrazol-4- yl)m...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576873((R)-4-(1-(2-Chloro-4- (((tetrahydro-2H-pyran-3- ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576874((S)-4-(1-(2-Chloro-4- (((tetrahydro-2H-pyran-3- ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576875(Ethyl 4-((3-chloro-4-(4- (5-cyano-2-((1- (methyl...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576876((+-)-4-(1-(2-Chloro-4- (((1- (methylsulfonyl) p...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576877(4-(1-(2-Chloro-4-(((2- (trifluoromethoxy)ethyl) ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576878(4-(1-(2-Chloro-4-(((2- (methylsulfonyl)ethyl) am...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576879(US11472791, Example 201)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576880(1-(4-(2-(((3R,4S)-1-((3- (Diethylamino)propyl) s...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576881(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-(pyrrolidin- 1...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576882(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-(piperidin-1- ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576883(1-(4-(2-(((3R,4S)-1-((3- (Dimethylamino)propyl) ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576884(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-((R)-3- methox...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576885(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-(4- methoxypip...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576886(1-(3-(((3R,4S)-3-Fluoro- 4-((4-(1-(2-hydroxy-2- ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576887(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-(4- methylpipe...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576888(1-(4-(2-(((3R,45)-1-((3- (4-Ethylpiperazin-1- yl...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576889(1-(4-(2-(((3R,4S)-3- Fluoro-1-((3-((1S,4S)-5- me...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576890(4-(3-(((3R,4S)-3-Fluoro- 4-((4-(1-(2-hydroxy-2- ...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576891(2-((1-((3- (Diethylamino)propyl) sulfonyl)piperi...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576892(4-(1-(2-Hydroxy-2- methylpropyl)-1H- pyrazol-4-y...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576893(4-(1-(2-Hydroxy-2- methylpropyl)-1H- pyrazol-4-y...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576894(2-((1-((4- (Diethylamino)butyl) sulfonyl)piperid...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576895(4-(1-(2-Hydroxy-2- methylpropyl)-1H- pyrazol-4-y...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576896(4-(1-(2-Hydroxy-2- methylpropyl)-1H- pyrazol-4-y...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM576897((S)-1-(4-(2-((1-((3-(3- Methoxypyrrolidin-1- yl)...)
Affinity DataIC50: <50nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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