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Found 268 with Last Name = 'fujio' and Initial = 'm'
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218398(CHEMBL1907861)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201292(7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyr...)
Affinity DataKi:  0.120nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218392(CHEMBL79277)
Affinity DataKi:  0.140nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218388(CHEMBL78986)
Affinity DataKi:  0.170nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218397(CHEMBL83611)
Affinity DataKi:  0.190nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201292(7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyr...)
Affinity DataKi:  0.220nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218396(CHEMBL315259)
Affinity DataKi:  0.240nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218397(CHEMBL83611)
Affinity DataKi:  0.320nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218399(CHEMBL79643)
Affinity DataKi:  0.440nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat striata 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50086855(CHEMBL82884 | Cyclohexanecarboxylic acid ((S)-1-ph...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50086855(CHEMBL82884 | Cyclohexanecarboxylic acid ((S)-1-ph...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat striata 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218400(CHEMBL1907669)
Affinity DataKi:  0.530nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50218391(CHEMBL79528)
Affinity DataKi:  0.550nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201280(CHEMBL394137 | {3-[(2-adamantan-1-yl-ethylamino)-m...)
Affinity DataKi:  0.660nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  0.780nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  1nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218395(CHEMBL311095)
Affinity DataKi:  1.10nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218393(CHEMBL79542)
Affinity DataKi:  1.10nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor from striata of wistar rats by [3H]- 8-OH -DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201280(CHEMBL394137 | {3-[(2-adamantan-1-yl-ethylamino)-m...)
Affinity DataKi:  1.5nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201277((4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][...)
Affinity DataKi:  1.80nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201292(7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyr...)
Affinity DataKi:  1.80nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201296(4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1...)
Affinity DataKi:  1.90nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201285(3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3...)
Affinity DataKi:  2nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201277((4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][...)
Affinity DataKi:  2.10nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201294(3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3...)
Affinity DataKi:  2.40nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201283(3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,...)
Affinity DataKi:  2.5nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201285(3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3...)
Affinity DataKi:  2.70nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201296(4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1...)
Affinity DataKi:  2.90nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218398(CHEMBL1907861)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]-Prazosin binding to Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201294(3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3...)
Affinity DataKi:  3.30nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  3.5nMAssay Description:Ability to displace [3H]-Prazosin binding to Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190677((R)-3'-(3-bromobenzo[b]thiophen-5-yl)spiro[1-azabi...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190686((R)-3'-(2,3-dimethylbenzo[b]thiophen-5-yl)spiro[1-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190696((2S)-3'-(5-bromothien-2-yl)-2'H-spiro[4-azabicyclo...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50164606((2R)-3'-(5-bromothien-2-yl)-2'H-spiro[4-azabicyclo...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to rat nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201299(7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4...)
Affinity DataKi:  4.20nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50086861(3-Methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat striata 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Welfide

Curated by ChEMBL
LigandPNGBDBM50086856(CHEMBL147279 | N-((S)-1-Phenethyl-pyrrolidin-2-ylm...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat striata 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201284(3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4...)
Affinity DataKi:  4.90nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201299(7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4...)
Affinity DataKi:  5.10nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Welfide

Curated by ChEMBL
LigandPNGBDBM50093797(Adamantane-1-carboxylic acid {1-[2-(4-cyano-phenyl...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201276(3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)me...)
Affinity DataKi:  5.80nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201280(CHEMBL394137 | {3-[(2-adamantan-1-yl-ethylamino)-m...)
Affinity DataKi:  5.90nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201287(CHEMBL435353 | N,N-dimethyl-3-((2-(tetrahydro-2H-p...)
Affinity DataKi:  6nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50201283(3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,...)
Affinity DataKi:  6.20nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50218396(CHEMBL315259)
Affinity DataKi:  6.40nMAssay Description:Ability to displace [3H]-Prazosin binding to Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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