TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK1 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK2 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of Ig-tagged human PD1/His-tagged human PDL1 interaction incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair