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Found 61 with Last Name = 'galineau' and Initial = 'l'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178936(2-(2-((dimethylamino)methyl)phenoxy)-5-methylbenze...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]paroxetine from SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50110788(2-(2-((dimethylamino)methyl)phenylthio)-5-methylan...)
Affinity DataKi:  1.65nMAssay Description:Displacement of [3H]paroxetine from SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178934(2-(2-((dimethylamino)methyl)phenylsulfinyl)-5-meth...)
Affinity DataKi:  4.15nMAssay Description:Displacement of [3H]paroxetine from SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178935(CHEMBL383422 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataKi:  10.3nMAssay Description:Displacement of [3H]paroxetine from SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183824(1-(2-bromobenzyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183823(1-(3-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  46nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183817(1-(2-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  47nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183813(1-benzyl-4-(4-phenylpiperazin-1-yl)piperidin-3-ol ...)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183818(1-(3-bromobenzyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183810(1-benzyl-3-(4-phenylpiperazin-1-yl)piperidin-4-ol ...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183825((E)-1-(3-iodoallyl)-4-(4-phenylpiperazin-1-yl)pipe...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183828(4-(4-phenylpiperazin-1-yl)piperidin-3-ol | CHEMBL3...)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183820((E)-1-(but-2-enyl)-3-(4-phenylpiperazin-1-yl)piper...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183814(3-(4-phenylpiperazin-1-yl)-1-(prop-2-ynyl)piperidi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178930((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178933(CHEMBL377714 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178931((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178932(CHEMBL204702 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183826((E)-1-(but-2-enyl)-4-(4-phenylpiperazin-1-yl)piper...)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183827((E)-1-(3-iodoallyl)-3-(4-phenylpiperazin-1-yl)pipe...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183816(3-(4-phenylpiperazin-1-yl)piperidin-4-ol | CHEMBL2...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183829(1-(4-bromobenzyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183809(1-allyl-4-(4-phenylpiperazin-1-yl)piperidin-3-ol |...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183821(1-allyl-3-(4-phenylpiperazin-1-yl)piperidin-4-ol |...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183819(1-(2-methylallyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178941(2-(2-((dimethylamino)methyl)phenylsulfonyl)-5-meth...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183822(1-(2-methylallyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50183812(1-(4-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178934(2-(2-((dimethylamino)methyl)phenylsulfinyl)-5-meth...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178939(2-((2-((dimethylamino)methyl)phenyl)(methoxy)methy...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178936(2-(2-((dimethylamino)methyl)phenoxy)-5-methylbenze...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178937(2'-Dimethylaminomethyl-5-methyl-biphenyl-2-ylamine...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178935(CHEMBL383422 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178938(CHEMBL381071 | N1-benzyl-N1-(2-((dimethylamino)met...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178937(2'-Dimethylaminomethyl-5-methyl-biphenyl-2-ylamine...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50110788(2-(2-((dimethylamino)methyl)phenylthio)-5-methylan...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178936(2-(2-((dimethylamino)methyl)phenoxy)-5-methylbenze...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178932(CHEMBL204702 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178930((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178940(CHEMBL205313 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178930((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178940(CHEMBL205313 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178933(CHEMBL377714 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178941(2-(2-((dimethylamino)methyl)phenylsulfonyl)-5-meth...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178938(CHEMBL381071 | N1-benzyl-N1-(2-((dimethylamino)met...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178939(2-((2-((dimethylamino)methyl)phenyl)(methoxy)methy...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178931((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178934(2-(2-((dimethylamino)methyl)phenylsulfinyl)-5-meth...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178931((2-amino-4-methylphenyl)(2-((dimethylamino)methyl)...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50178940(CHEMBL205313 | N1-(2-((dimethylamino)methyl)phenyl...)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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