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Found 277 with Last Name = 'georgey' and Initial = 'hh'
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567652(CHEMBL4878693)
Affinity DataKi:  25nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) after 10 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567655(CHEMBL4873710)
Affinity DataKi:  25nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) after 10 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567666(CHEMBL4850615)
Affinity DataKi:  40nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) after 10 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567666(CHEMBL4850615)
Affinity DataKi:  127nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567665(CHEMBL4855877)
Affinity DataKi:  131nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) after 10 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567666(CHEMBL4850615)
Affinity DataKi:  144nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567665(CHEMBL4855877)
Affinity DataKi:  203nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567652(CHEMBL4878693)
Affinity DataKi:  208nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567665(CHEMBL4855877)
Affinity DataKi:  437nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567652(CHEMBL4878693)
Affinity DataKi:  581nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567655(CHEMBL4873710)
Affinity DataKi:  823nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567655(CHEMBL4873710)
Affinity DataKi:  1.27E+3nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567655(CHEMBL4873710)
Affinity DataKi:  3.78E+3nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567652(CHEMBL4878693)
Affinity DataKi:  9.12E+3nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567665(CHEMBL4855877)
Affinity DataKi:  1.16E+4nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50567666(CHEMBL4850615)
Affinity DataKi:  5.69E+4nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089076(CHEMBL3577642)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50347388(CHEMBL1234833)
Affinity DataIC50:  3nMAssay Description:Inhibition of human CDK2 expressed in baculovirus infected Sf9 cells using Histone H1 as substrate incubated for 10 mins by scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088896(CHEMBL3577645)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088857(CHEMBL3577567)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant COX-2 using arachidonic acid as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50578582(CHEMBL4849659)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant COX-2 using arachidonic acid as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50:  7nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Bos taurus (Cattle))
Future University

LigandPNGBDBM226165(N'-[4-Methoxybenzylidene-2-(6-chloro)-3-(4-met...)
Affinity DataIC50:  10nMpH: 7.4 T: 2°CAssay Description:The assay mixture contained 50 μM Tris-HCl buffer (pH 7.4), 50 μM NADPH, 10 μl DMSO or the same volume of DMSO solution containing the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Cairo University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50578584(CHEMBL4874336)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant COX-2 using arachidonic acid as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  18nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088859(CHEMBL3577565)
Affinity DataIC50:  20nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50:  21nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50:  21nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089082(CHEMBL3577636)
Affinity DataIC50:  23nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50:  23nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089082(CHEMBL3577636)
Affinity DataIC50:  23nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089081(CHEMBL3577637)
Affinity DataIC50:  23nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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