TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: >0.0480nMAssay Description:Binding affinity to human adenosine A2a receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.420nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.610nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.630nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 0.890nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.07nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.39nMAssay Description:Binding affinity towards human cloned 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.44nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.45nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.48nMAssay Description:Binding affinity towards human cloned 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.51nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.76nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.29nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.47nMAssay Description:Binding affinity towards human cloned 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.59nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.92nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.99nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 3.29nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 3.44nMAssay Description:Binding affinity towards human cloned 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 3.77nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair