Compile Data Set for Download or QSAR
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Found 61 with Last Name = 'gorczynski' and Initial = 'mj'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295043((E)-12-Nitrooctadec-12-enoic Acid | CHEMBL549351)
Affinity DataIC50:  39nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295044((E)-13-Nitrooctadec-12-enoic Acid | CHEMBL540732)
Affinity DataIC50:  190nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataIC50:  250nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataIC50:  410nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295046((E)-10-Nitrohexadec-9-enoic Acid | CHEMBL564368)
Affinity DataIC50:  630nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31183(thiazol-2-amine, 14)
Affinity DataIC50:  700nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295047((E)-9-Nitrohexadec-9-enoicAcid | CHEMBL560513)
Affinity DataIC50:  830nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | CHEMBL550762 | N...)
Affinity DataIC50:  980nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295044((E)-13-Nitrooctadec-12-enoic Acid | CHEMBL540732)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31183(thiazol-2-amine, 14)
Affinity DataIC50:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295043((E)-12-Nitrooctadec-12-enoic Acid | CHEMBL549351)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295049((E)-10-nitrooctadec-9-enoic acid | CHEMBL561371)
Affinity DataIC50:  1.61E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295050((E)-5-Nitrooctadec-5-enoic Acid | CHEMBL561776)
Affinity DataIC50:  1.68E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295051((E)-6-Nitrooctadec-5-enoic Acid | CHEMBL569372)
Affinity DataIC50:  1.72E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31175(thiazol-2-amine, 5)
Affinity DataIC50:  3.00E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31185(thiazol-2-amine, 17)
Affinity DataIC50:  3.20E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31186(thiazol-2-amine, 18)
Affinity DataIC50:  3.20E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31182(thiazol-2-amine, 13)
Affinity DataIC50:  3.30E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31185(thiazol-2-amine, 17)
Affinity DataIC50:  3.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31182(thiazol-2-amine, 13)
Affinity DataIC50:  5.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31179(thiazol-2-amine, 9)
Affinity DataIC50:  6.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31178(thiazol-2-amine, 8)
Affinity DataIC50:  6.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31175(thiazol-2-amine, 5)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31178(thiazol-2-amine, 8)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataIC50:  9.60E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31179(thiazol-2-amine, 9)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31176(thiazol-2-amine, 6)
Affinity DataIC50:  1.20E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | CHEMBL550762 | N...)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295049((E)-10-nitrooctadec-9-enoic acid | CHEMBL561371)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295047((E)-9-Nitrohexadec-9-enoicAcid | CHEMBL560513)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295046((E)-10-Nitrohexadec-9-enoic Acid | CHEMBL564368)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295050((E)-5-Nitrooctadec-5-enoic Acid | CHEMBL561776)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295051((E)-6-Nitrooctadec-5-enoic Acid | CHEMBL569372)
Affinity DataIC50: >1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31187(thiazol-2-amine, 19)
Affinity DataIC50:  1.65E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31188(thiazol-2-amine, 20)
Affinity DataIC50:  1.70E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31188(thiazol-2-amine, 20)
Affinity DataIC50:  1.80E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31177(thiazol-2-amine, 7)
Affinity DataIC50:  1.80E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31176(thiazol-2-amine, 6)
Affinity DataIC50:  1.85E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31184(thiazol-2-amine, 16)
Affinity DataIC50:  2.05E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31181(thiazol-2-amine, 11)
Affinity DataIC50:  2.25E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31186(thiazol-2-amine, 18)
Affinity DataIC50:  2.35E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31180(thiazol-2-amine, 10)
Affinity DataIC50:  3.60E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31177(thiazol-2-amine, 7)
Affinity DataIC50:  4.05E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31184(thiazol-2-amine, 16)
Affinity DataIC50:  4.90E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31181(thiazol-2-amine, 11)
Affinity DataIC50:  6.10E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31187(thiazol-2-amine, 19)
Affinity DataIC50:  6.60E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31180(thiazol-2-amine, 10)
Affinity DataIC50:  1.10E+5nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31189(thiazol-2-amine, 21)
Affinity DataIC50: >5.00E+5nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

LigandPNGBDBM31189(thiazol-2-amine, 21)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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