Affinity DataIC50: 0.130nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivation relative to Org 31710More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivation relative to Org 31710More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.610nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.980nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.14nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.25nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.64nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.89nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 8.48nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 133nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 193nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 314nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 318nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 598nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.810nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.45E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.34E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10.6nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.960nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10.3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 258nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 198nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 513nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair