Compile Data Set for Download or QSAR
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Found 76 with Last Name = 'hamersma' and Initial = 'h'
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375439(CHEMBL410304)
Affinity DataIC50:  0.130nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375445(CHEMBL445946)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivation relative to Org 31710More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375444(CHEMBL258861)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivation relative to Org 31710More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375424(ULIPRISTAL ACETATE | Ulipristal)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375438(CHEMBL410923)
Affinity DataIC50:  0.270nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375425(CHEMBL259879)
Affinity DataIC50:  0.330nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375440(CHEMBL411522)
Affinity DataIC50:  0.430nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375433(CHEMBL258522)
Affinity DataIC50:  0.470nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375441(CHEMBL260330)
Affinity DataIC50:  0.550nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375442(CHEMBL260764)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375437(CHEMBL409661)
Affinity DataIC50:  0.610nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375436(CHEMBL260869)
Affinity DataIC50:  0.630nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375443(CHEMBL408424)
Affinity DataIC50:  0.75nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375434(CHEMBL407371)
Affinity DataIC50:  0.980nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375427(CHEMBL411086)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375430(CHEMBL409905)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375426(CHEMBL268788)
Affinity DataIC50:  3.14nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375428(CHEMBL411063)
Affinity DataIC50:  3.25nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375429(CHEMBL438593)
Affinity DataIC50:  3.64nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233026(CHEMBL403138 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375435(CHEMBL406439)
Affinity DataIC50:  7.89nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375432(CHEMBL258521)
Affinity DataIC50:  8.48nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375431(CHEMBL261650)
Affinity DataIC50:  14.8nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(CHEMBL403139 | N-((1S,13bR)-6-chloro-1,2,3,4,9,13b...)
Affinity DataIC50:  26nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233014((rac)-N-(6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4a...)
Affinity DataIC50:  43nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233013(CHEMBL253944 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  133nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233009(CHEMBL253734 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  193nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233028(1-((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-ox...)
Affinity DataIC50:  314nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233020(CHEMBL252451 | N-((1S,13bR)-6,7-dichloro-1,3,4,13b...)
Affinity DataIC50:  318nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataIC50:  730nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233015(CHEMBL252646 | N-((1S,13bR)-7-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233006(((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-...)
Affinity DataEC50:  598nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(CHEMBL403139 | N-((1S,13bR)-6-chloro-1,2,3,4,9,13b...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233008(2,2,2-trifluoro-N-((1S,13bR)-5-vinyl-1,3,4,13b-tet...)
Affinity DataEC50:  0.810nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233009(CHEMBL253734 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  4.45E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233012(CHEMBL252449 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233010(CHEMBL252253 | N-((1R,13bS)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233011(((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-...)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233014((rac)-N-(6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4a...)
Affinity DataEC50:  10.6nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233017(CHEMBL252850 | N-((1S,13bR)-5-acetyl-1,3,4,13b-tet...)
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233016(CHEMBL253735 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233018(CHEMBL401627 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233013(CHEMBL253944 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  10.3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233019(CHEMBL402526 | N-((1S,13bR)-5-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233021(CHEMBL252648 | N-((1S,13bR)-6-acetyl-1,3,4,13b-tet...)
Affinity DataEC50:  258nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233023(CHEMBL404432 | N-((1S,13bR)-6-chloro-9-methyl-1,2,...)
Affinity DataEC50:  9.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233025(CHEMBL404433 | N-((1S,13bR)-5,6-dichloro-1,3,4,13b...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataEC50:  198nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233024((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4...)
Affinity DataEC50:  513nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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