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Found 120 with Last Name = 'hansen' and Initial = 'tv'
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338500((S)-1-((1-benzyl-1H-1,2,3-triazol-5-yl)methyl)-5-(...)
Affinity DataKi:  10.5nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338491((S)-1-((1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1H...)
Affinity DataKi:  14.5nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50273338((S)-1-((1-(2-Fluoroethyl)-1H-[1,2,3]-triazol-4-yl)...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(CHEMBL598608 | GSK-3787)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 24 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338500((S)-1-((1-benzyl-1H-1,2,3-triazol-5-yl)methyl)-5-(...)
Affinity DataIC50:  9nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50273337((S)-1-((1-(2-Fluoroethyl)-1H-[1,2,3]-triazol-4-yl)...)
Affinity DataIC50:  16.7nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338491((S)-1-((1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1H...)
Affinity DataIC50:  17nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338489((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  18nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338488((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  21nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338486((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  21nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338487((S)-1-((1-(biphenyl-4-yl)-1H-1,2,3-triazol-4-yl)me...)
Affinity DataIC50:  23nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  29nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 40 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  30nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 40 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338492((S)-1-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)-5-(...)
Affinity DataIC50:  30nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM10318((S)-5-{1-[2-(Phenoxymethyl)pyrrolidinyl]sulfonyl}i...)
Affinity DataIC50:  44nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338490((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  44nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338498((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  70nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338494((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  103nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM10305((S)-5-[1-(2-Methoxymethyl)pyrrolidinylsulfonyl]isa...)
Affinity DataIC50:  120nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338495((S)-1-((1-(biphenyl-4-yl)-1H-1,2,3-triazol-5-yl)me...)
Affinity DataIC50:  136nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338499((S)-1-((1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1H...)
Affinity DataIC50:  136nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataIC50:  155nMAssay Description:Binding affinity to N-terminal hexa-histidine tagged and fluorescein-labeled human PPAR-beta/delta (164 to 441 residues) expressed in Escherichia col...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338501((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  207nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338496((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  213nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134238(CHEMBL3740002)
Affinity DataIC50:  241nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 24 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338493((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  243nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50338497((S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1...)
Affinity DataIC50:  267nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  284nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(CHEMBL598608 | GSK-3787)
Affinity DataIC50:  284nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  301nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  423nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50:  598nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  600nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  600nMAssay Description:Inhibition of pig brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  600nMAssay Description:Inhibition of pig tubulin polymerizationMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(CHEMBL598608 | GSK-3787)
Affinity DataIC50:  648nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50:  907nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  949nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM22817(5-nitro-2,3-dihydro-1H-indole-2,3-dione | CHEMBL11...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of caspase 3 using Ac-DEVD-AFC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(CHEMBL598608 | GSK-3787)
Affinity DataIC50:  1.32E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134238(CHEMBL3740002)
Affinity DataIC50:  1.43E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134239(CHEMBL3740264)
Affinity DataIC50:  1.93E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056777(CHEMBL3331358)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50060957(2-Hydroxyestradol 2-methyl ether | 2-methoxy-17bet...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056783(CHEMBL3331351)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056779(CHEMBL3331356)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056782(CHEMBL3331353)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056775(CHEMBL3331360)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50056798(CHEMBL3331347)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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