TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110delta using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110delta using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110delta using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110gamma using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110gamma using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110gamma using [32P]ATP after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of recombinant GST-tagged PI3K p110alpha by KinaseGlo assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair