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Found 194 with Last Name = 'ilas' and Initial = 'j'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of [3H]CCPA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261591(3-(Benzyl(2-(4-carbamimidoylbenzyl)-4-methyl-3-oxo...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261568(CHEMBL468812 | Methyl 3-(benzyl(2-(4-carbamimidoyl...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261566(CHEMBL468642 | Ethyl 2-(Benzyl(2-(4-carbamimidoylb...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370631(CHEMBL607303)
Affinity DataKi:  5.47nMAssay Description:Inhibition of [3H]CCPA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261592(CHEMBL468340 | Ethyl 4-(benzyl(2-(4-carbamimidoylb...)
Affinity DataKi:  5.80nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261593(4-(Benzyl(2-(4-carbamimidoylbenzyl)-4-methyl-3-oxo...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370629(CHEMBL607302)
Affinity DataKi:  8.23nMAssay Description:Inhibition of [3H]CCPA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50163564(3-Benzyl-8-cyclopentyl-1-propyl-3,7-dihydro-purine...)
Affinity DataKi:  8.70nMAssay Description:Inhibition of [3H]R-PIA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261567(2-(Benzyl(2-(4-carbamimidoylbenzyl)-4-methyl-3-oxo...)
Affinity DataKi:  11nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370632(CHEMBL607025)
Affinity DataKi:  15.7nMAssay Description:Inhibition of [3H]CCPA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147480(CHEMBL109999 | N-(3-Amino-2-imino-2,3,4,5,6,7-hexa...)
Affinity DataKi:  22nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253900(CHEMBL468464 | Ethyl 4-({2-[(4-carbamimidoylphenox...)
Affinity DataKi:  25nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147477(CHEMBL111122 | N-(3-Amino-2-imino-2,3,4,5,6,7-hexa...)
Affinity DataKi:  42nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370630(CHEMBL607024)
Affinity DataKi:  45nMAssay Description:Percent inhibition of [3H]PSB-11 binding to adenosine A3 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370632(CHEMBL607025)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]PSB-298 binding to adenosine A2b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  51nMAssay Description:Inhibition of [3H]ZM-241,385 binding to adenosine A2b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50163564(3-Benzyl-8-cyclopentyl-1-propyl-3,7-dihydro-purine...)
Affinity DataKi:  54.6nMAssay Description:Inhibition of [3H]PSB-11 binding to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253860(CHEMBL513670 | Ethyl 4-(Benzyl{2-[(4-carbamimidoyl...)
Affinity DataKi:  60nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147489(CHEMBL109696 | N-((R)-2-Amino-4,5,6,7-tetrahydro-b...)
Affinity DataKi:  71nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147475(CHEMBL419008 | N-((R)-2-Amino-4,5,6,7-tetrahydro-b...)
Affinity DataKi:  77nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147487(CHEMBL111160 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147488(CHEMBL110201 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147485(2-(6-Methyl-2-oxo-3-p-tolylmethanesulfonylamino-2H...)
Affinity DataKi:  102nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253817(CHEMBL460144 | Ethyl 2-(benzyl{2-[(4-carbamimidoyl...)
Affinity DataKi:  110nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147483(CHEMBL327136 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147476(2-[3-(4-Fluoro-phenylmethanesulfonylamino)-6-methy...)
Affinity DataKi:  149nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253932(CHEMBL459318 | Ethyl 2-(N-{2-[(4-carbamimidoylphen...)
Affinity DataKi:  156nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147490(CHEMBL111468 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  157nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147486(2-[3-(2-Chloro-4-fluoro-phenylmethanesulfonylamino...)
Affinity DataKi:  157nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370630(CHEMBL607024)
Affinity DataKi:  160nMAssay Description:Inhibition of [3H]CCPA binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132525(2-(6-Methyl-2-oxo-3-phenylmethanesulfonylamino-2H-...)
Affinity DataKi:  170nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50165956((S)-2-{2-[4-(4-Carbamimidoyl-benzyl)-3-oxo-3,4-dih...)
Affinity DataKi:  206nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253858(CHEMBL461210 | Ethyl 2-(benzyl{2-[(4-carbamimidoyl...)
Affinity DataKi:  320nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370632(CHEMBL607025)
Affinity DataKi:  350nMAssay Description:Inhibition of [3H]PSB-11 binding to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253818(2-(Benzyl{2-[(4-carbamimidoylphenoxy)methyl]-2,4-d...)
Affinity DataKi:  377nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253780(CHEMBL517875 | Ethyl 2-(benzyl{2-[(4-carbamimidoyl...)
Affinity DataKi:  380nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  470nMAssay Description:Inhibition of [3H]MSX-2 binding to adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253898(4-(Benzyl{2-[(4-carbamimidoylphenoxy)methyl]-2,4-d...)
Affinity DataKi:  490nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50163564(3-Benzyl-8-cyclopentyl-1-propyl-3,7-dihydro-purine...)
Affinity DataKi:  511nMAssay Description:Inhibition of [3H]NECA binding to adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147479(2-[6-Methyl-2-oxo-3-(3-trifluoromethyl-phenylmetha...)
Affinity DataKi:  562nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147478(CHEMBL109217 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  652nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253899(CHEMBL512630 | Ethyl 4-(benzyl{2-[(4-carbamimidoyl...)
Affinity DataKi:  670nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  759nMAssay Description:Inhibition of [3H]PSB-11 binding to adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50253859(2-(Benzyl{2-[(4-carbamimidoylphenoxy)methyl]-2,4-d...)
Affinity DataKi:  879nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50165952(2-Benzyl-N-[4-(4-carbamimidoyl-benzyl)-3-oxo-3,4-d...)
Affinity DataKi:  973nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370631(CHEMBL607303)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]PSB-298 binding to adenosine A2b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50261592(CHEMBL468340 | Ethyl 4-(benzyl(2-(4-carbamimidoylb...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50147492(CHEMBL109345 | N-((S)-2-Amino-4,5,6,7-tetrahydro-b...)
Affinity DataKi:  1.16E+3nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50370632(CHEMBL607025)
Affinity DataKi:  1.27E+3nMAssay Description:Inhibition of [3H]MSX-2 binding to adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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