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Found 59 with Last Name = 'kandalkar' and Initial = 'sr'
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451174(CHEMBL4202457)
Affinity DataKi:  0.600nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451177(CHEMBL4210264)
Affinity DataKi:  1.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451169(CHEMBL4207346)
Affinity DataKi:  1.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451139(CHEMBL4204605)
Affinity DataKi:  1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451140(CHEMBL4216271)
Affinity DataKi:  1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451167(CHEMBL4206823)
Affinity DataKi:  1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451164(CHEMBL4208941)
Affinity DataKi:  1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451168(CHEMBL4211702)
Affinity DataKi:  2.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM28393((+)-EHNA | (2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451138(CHEMBL4203116)
Affinity DataKi:  2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451173(CHEMBL4214254)
Affinity DataKi:  2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451165(CHEMBL4204068)
Affinity DataKi:  2.30nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451166(CHEMBL4209345)
Affinity DataKi:  2.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451141(CHEMBL4216791)
Affinity DataKi:  2.70nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451142(CHEMBL4211824)
Affinity DataKi:  2.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451158(CHEMBL4218202)
Affinity DataKi:  4.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451171(CHEMBL4214511)
Affinity DataKi:  5.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451178(CHEMBL4203469)
Affinity DataKi:  5.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451170(CHEMBL4214658)
Affinity DataKi:  6.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451133(CHEMBL4218610)
Affinity DataKi:  25nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451172(CHEMBL4215142)
Affinity DataKi:  29nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451134(CHEMBL4206867)
Affinity DataKi:  49nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451159(CHEMBL4205307)
Affinity DataKi:  53nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451137(CHEMBL4207993)
Affinity DataKi:  54nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451135(CHEMBL4206350)
Affinity DataKi:  66nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451100(CHEMBL4208733)
Affinity DataKi:  69nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50451136(CHEMBL4211238)
Affinity DataKi:  135nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382410(CHEMBL2022568)
Affinity DataIC50:  910nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382411(CHEMBL2022569)
Affinity DataIC50:  4.27E+3nMAssay Description:Inhibition of rat His6-tagged Hao2 expressed in Escherichia coli BL21/DE3 using 2-hydroxyoctanoic acid as substrate measured every 10 secs by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382413(CHEMBL2022571)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382412(CHEMBL2022570)
Affinity DataIC50:  4.57E+4nMAssay Description:Inhibition of rat His6-tagged Hao1 expressed in Escherichia coli BL21/DE3 using glcolic acid as substrate measured every 10 secs by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615265(CHEMBL5276863)
Affinity DataEC50:  450nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615266(CHEMBL5279712)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615267(CHEMBL5288503)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615268(CHEMBL5290142)
Affinity DataEC50:  2.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615269(CHEMBL5267943)
Affinity DataEC50:  34nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615264(CHEMBL5288114)
Affinity DataEC50:  400nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615263(CHEMBL5275999)
Affinity DataEC50:  2.73E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHexokinase-4(Homo sapiens (Human))TBA
LigandPNGBDBM50615262(CHEMBL5282187)
Affinity DataEC50:  310nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
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