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Found 66 with Last Name = 'kikuchi' and Initial = 't'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  18.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  19.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  46.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM11638(CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50437871(CHEMBL2407927)
Affinity DataKi:  2.00E+8nMAssay Description:Inhibition of ALAD (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043326(CHEMBL438733 | c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-...)
Affinity DataIC50:  0.0930nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataIC50:  0.120nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataIC50:  0.150nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368776(CHEMBL1790962)
Affinity DataIC50:  0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043322(CHEMBL427748 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368773(CHEMBL1790959)
Affinity DataIC50:  0.180nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368774(CHEMBL1790963)
Affinity DataIC50:  0.190nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368775(CHEMBL1790960)
Affinity DataIC50:  0.200nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368772(CHEMBL2373291)
Affinity DataIC50:  0.25nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368774(CHEMBL1790963)
Affinity DataIC50:  0.330nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368777(CHEMBL2373292)
Affinity DataIC50:  0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368776(CHEMBL1790962)
Affinity DataIC50:  0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043324(CHEMBL411171 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  0.450nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368772(CHEMBL2373291)
Affinity DataIC50:  0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368777(CHEMBL2373292)
Affinity DataIC50:  0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043322(CHEMBL427748 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  0.75nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043326(CHEMBL438733 | c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-...)
Affinity DataIC50:  5.90nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043324(CHEMBL411171 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  8.60nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084312((+)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(2-prope...)
Affinity DataIC50:  50nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes (high)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084320(5-Chloro-1-{3-[4-(3-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataIC50:  130nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084310(1-{3-[4-(3-Bromo-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  150nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50369619(CHEMBL1743967)
Affinity DataIC50:  240nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084307(1-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  260nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084325(5-Chloro-1-{3-[4-(3-propoxy-phenyl)-piperazin-1-yl...)
Affinity DataIC50:  370nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084313(5-Chloro-1-{3-[4-(3-nitro-phenyl)-piperazin-1-yl]-...)
Affinity DataIC50:  390nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM81982(CAS_97-39-2 | DITOLYLGUANIDINE | DTG | Di-o-tolylg...)
Affinity DataIC50:  400nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084308(1-{3-[4-(3-Bromo-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  420nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084324(1-{3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  460nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084311(5-Methoxy-1-{3-[4-(3-trifluoromethyl-phenyl)-piper...)
Affinity DataIC50:  490nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084321(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  600nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084326(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  620nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084329(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  650nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084323(CHEMBL299492 | N-(3-{4-[3-(5-Chloro-2-oxo-3,4-dihy...)
Affinity DataIC50:  670nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084319(1-{3-[4-(3-Amino-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  710nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084315(1-{3-[4-(3-Hydroxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataIC50:  810nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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