Compile Data Set for Download or QSAR
maximum 50k data
Found 56 with Last Name = 'koukoulitsa' and Initial = 'c'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490702(CHEMBL2337686)
Affinity DataIC50:  0.347nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490707(CHEMBL2337687)
Affinity DataIC50:  0.912nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490709(CHEMBL2337688)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490706(CHEMBL2337677)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  7nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490699(CHEMBL2337681)
Affinity DataIC50:  43nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM16312((4S)-6-fluoro-2,3-dihydrospiro[1-benzopyran-4,4'-i...)
Affinity DataIC50:  70nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM16312((4S)-6-fluoro-2,3-dihydrospiro[1-benzopyran-4,4'-i...)
Affinity DataIC50:  249nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM16312((4S)-6-fluoro-2,3-dihydrospiro[1-benzopyran-4,4'-i...)
Affinity DataIC50:  250nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490704(CHEMBL2337684)
Affinity DataIC50:  331nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336704((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-2-yl)(...)
Affinity DataIC50:  390nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336708((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl)(...)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490698(CHEMBL2337683)
Affinity DataIC50:  417nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490708(CHEMBL2337685)
Affinity DataIC50:  501nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490701(CHEMBL2337679)
Affinity DataIC50:  708nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016389(CHEMBL3264340)
Affinity DataIC50:  740nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50237838((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(4,5-dihy...)
Affinity DataIC50:  741nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490703(CHEMBL2337678)
Affinity DataIC50:  832nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336705((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-2-yl)(...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336703((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-2-yl)(...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336702(CHEMBL1673033 | [1-(2,4-Difluoro-3-hydroxyphenyl)-...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490705(CHEMBL2337682)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50:  1.84E+3nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50146187((3-Benzoyl-pyrrol-1-yl)-acetic acid | 2-(3-benzoyl...)
Affinity DataIC50:  1.97E+3nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016391(CHEMBL3264344)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50133496((2R)-3-(3,4-dihydroxyphenyl)-2-[(2E)-3-(3,4-dihydr...)
Affinity DataIC50:  3.91E+3nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016386(CHEMBL3264336)
Affinity DataIC50:  5.26E+3nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50308548(4-(3-Benzoyl-1H-pyrrol-1-yl)butanoic acid | CHEMBL...)
Affinity DataIC50:  6.04E+3nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Patras

Curated by ChEMBL
LigandPNGBDBM50490700(CHEMBL2337680)
Affinity DataIC50:  6.46E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016384(CHEMBL3264333)
Affinity DataIC50: >7.50E+3nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50308547(3-(3-Benzoyl-1H-pyrrol-1-yl)propanoic acid | CHEMB...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336706((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl)(...)
Affinity DataIC50:  9.93E+3nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016396(CHEMBL3264352)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016395(CHEMBL3264351)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50308549(1-(2H-Tetrazole-5-yl)-1H-pyrrol-3-yl)(phenyl)metha...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016399(CHEMBL3264655)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016397(CHEMBL3264654)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016394(CHEMBL3264350)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016393(CHEMBL3264346)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016392(CHEMBL3264345)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016390(CHEMBL3264343)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016387(CHEMBL3264338)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016383(CHEMBL3264327)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016382(CHEMBL3264326)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016381(CHEMBL3264324)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016380(CHEMBL3264323)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Ratka Resanovica1

Curated by ChEMBL
LigandPNGBDBM50016379(CHEMBL3264322)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of horse serum BChE using butyrylthiocholine iodide as substrate preincubated for 35 mins followed by enzyme addition measured after 3 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50308550(1-(2H-tetrazole-5-yl)-1H-pyrrol-2-yl)(phenyl)metha...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of aldose reductase in Fischer-344 rat lens homogenate by spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Aristotle University Of Thessaloniki

Curated by ChEMBL
LigandPNGBDBM50336707((1-(3,5-Difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl)(...)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of rat lens ALR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: