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Found 62 with Last Name = 'leou' and Initial = 'js'
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of Aurora B kinaseMore data for this Ligand-Target Pair
TargetAurora kinase C(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of Aurora C kinaseMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  13nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase C(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  61nMAssay Description:Inhibition of Aurora C kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  79nMAssay Description:Inhibition of Aurora B kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)
Affinity DataIC50:  7nMAssay Description:Inhibition of GST-tagged EGFR expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of GST-tagged EGFR expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  20nMAssay Description:Inhibition of GST-tagged EGFR expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479526(CHEMBL515560)
Affinity DataIC50:  33nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322816(1-{4-[2-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-ylamin...)
Affinity DataIC50:  43nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322821((S)-N-(4-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)
Affinity DataIC50:  82nMAssay Description:Inhibition of GST-tagged EGFR expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322820(CHEMBL1172781 | S-2-(5,6-Diphenylfuro[2,3-d]pyrimi...)
Affinity DataIC50:  223nMAssay Description:Inhibition of GST-tagged EGFR expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322805((5,6-Diphenylfuro[2,3-d]pyrimidin-4-yl)-[2-(1H-imi...)
Affinity DataIC50:  296nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322817(CHEMBL1173801 | N-{4-[2-(5,6-Diphenylfuro[2,3-d]py...)
Affinity DataIC50:  304nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM14800(2-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-et...)
Affinity DataIC50:  309nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322812(4-(3,5-Dimethylpiperazin-1-yl)-5,6-diphenylfuro[2,...)
Affinity DataIC50:  334nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479524(CHEMBL474344)
Affinity DataIC50:  449nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479510(CHEMBL515112)
Affinity DataIC50:  460nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322810((5,6-Diphenylfuro[2,3-d]pyrimidin-4-yl)-(2-pyridin...)
Affinity DataIC50:  535nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322813(4-[2-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-ylamino)e...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322807(CHEMBL1173151 | [2-(4-Aminophenyl)ethyl]-(5,6-diph...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479520(CHEMBL473334)
Affinity DataIC50:  719nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322809(2-[2-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-ylamino)e...)
Affinity DataIC50:  760nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322808(CHEMBL1173152 | S-2-(5,6-Diphenylfuro[2,3-d]pyrimi...)
Affinity DataIC50:  792nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322806(3-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-ylamino)prop...)
Affinity DataIC50:  796nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479527(CHEMBL461954)
Affinity DataIC50:  804nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322803(1-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-yl)piperidin...)
Affinity DataIC50:  807nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322811((2,5-Dimethoxy-2,5-dihydrofuran-2-ylmethyl)-(5,6-d...)
Affinity DataIC50:  827nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479521(CHEMBL461785)
Affinity DataIC50:  838nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322815((4-Aminobenzyl)-(5,6-diphenylfuro[2,3-d]pyrimidin-...)
Affinity DataIC50:  945nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479522(CHEMBL473131)
Affinity DataIC50:  960nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322814(1-(5,6-Diphenylfuro[2,3-d]pyrimidin-4-ylamino)prop...)
Affinity DataIC50:  973nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479528(CHEMBL518032)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479511(CHEMBL474540)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479517(CHEMBL461599)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479525(CHEMBL473333)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479531(CHEMBL517573)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479512(CHEMBL516353)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479529(CHEMBL514951)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479516(CHEMBL460720)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479519(CHEMBL461784)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479513(CHEMBL460905)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322804((5,6-Diphenylfuro[2,3-d]pyrimidin-4-yl)-(2-morphol...)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479533(CHEMBL460728)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479518(CHEMBL461972)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479509(CHEMBL473948)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50322802((5,6-Diphenylfuro[2,3-d]pyrimidin-4-yl)-(3-imidazo...)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of Aurora AChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479530(CHEMBL517571)
Affinity DataIC50:  5.25E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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