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Found 122 with Last Name = 'martasek' and Initial = 'p'
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061231(2-Amino-5-(N'-propyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  1.80nMAssay Description:Compound was tested for binding affinity against recombinant inducible nitric oxide synthase (iNOS) from mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061231(2-Amino-5-(N'-propyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  57nMAssay Description:Compound was tested for binding affinity against neuronal nitric oxide synthase(nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50196043(3-N-(L-ArgNO2)-trans-3-amino-L-proline-NH2 ditrifl...)
Affinity DataKi:  87nMAssay Description:Inhibition of rat nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21962(3-[(4S)-4-amino-5-[(2-aminoethyl)(hydroxy)amino]pe...)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM22030((2S)-2-amino-N-[(1S)-3-amino-1-(aminocarbonyl)prop...)
Affinity DataKi:  130nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21960(3-[(4S)-4-amino-5-[(2-aminoethyl)amino]pentyl]-1-n...)
Affinity DataKi:  170nM ΔG°:  -39.3kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061230(1-Acetyl-4-(N'-allyl-guanidino)-butyl-ammonium)
Affinity DataKi:  200nMAssay Description:Compound was tested for binding affinity against neuronal nitric oxide synthase(nNOS)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21964((2S,4R)-4-[(2S)-2-amino-N-hydroxy-5-(1-nitrocarbam...)
Affinity DataKi:  310nM ΔG°:  -37.8kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369442(CHEMBL1202118)
Affinity DataKi:  320nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50196042(4-N-(L-ArgNO2)-Nalpha-benzyl-trans-4-amino-L-proli...)
Affinity DataKi:  328nMAssay Description:Inhibition of rat nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369441(CHEMBL1202106)
Affinity DataKi:  330nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21961((2S,4R)-4-[(2S)-2-amino-5-(1-nitrocarbamimidamido)...)
Affinity DataKi:  330nM ΔG°:  -37.6kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061232(2-Amino-5-(N'-prop-2-ynyl-guanidino)-pentanoic aci...)
Affinity DataKi:  430nMAssay Description:Compound was tested for binding affinity against neuronal nitric oxide synthase(nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369436(CHEMBL1204423)
Affinity DataKi:  450nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21963(3-[(4S)-4-amino-5-[1-(2-aminoethyl)hydrazin-1-yl]p...)
Affinity DataKi:  560nM ΔG°:  -36.3kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50225106((2S)-2-amino-5-{[(E)-amino(nitroimino)methyl]amino...)
Affinity DataKi:  610nM ΔG°:  -36.1kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061232(2-Amino-5-(N'-prop-2-ynyl-guanidino)-pentanoic aci...)
Affinity DataKi:  620nMAssay Description:Compound was tested for binding affinity against recombinant inducible nitric oxide synthase (iNOS) from mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50225106((2S)-2-amino-5-{[(E)-amino(nitroimino)methyl]amino...)
Affinity DataKi:  720nM ΔG°:  -35.6kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369440(CHEMBL1202117)
Affinity DataKi:  770nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50061232(2-Amino-5-(N'-prop-2-ynyl-guanidino)-pentanoic aci...)
Affinity DataKi:  810nMAssay Description:Compound was tested for binding affinity against Endothelial nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369437(CHEMBL1204426)
Affinity DataKi:  1.10E+3nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369438(CHEMBL1202116)
Affinity DataKi:  1.70E+3nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369301(CHEMBL1788374)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of Neuronal Nitric oxide synthase enzyme (nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369303(CHEMBL1204422)
Affinity DataKi:  2.00E+3nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against bovine brain nNOS (Neuronal nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061230(1-Acetyl-4-(N'-allyl-guanidino)-butyl-ammonium)
Affinity DataKi:  2.10E+3nMAssay Description:Compound was tested for binding affinity against recombinant inducible nitric oxide synthase (iNOS) from mouseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50061230(1-Acetyl-4-(N'-allyl-guanidino)-butyl-ammonium)
Affinity DataKi:  3.10E+3nMAssay Description:Compound was tested for binding affinity against Endothelial nitric oxide synthaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50225106((2S)-2-amino-5-{[(E)-amino(nitroimino)methyl]amino...)
Affinity DataKi:  4.28E+3nM ΔG°:  -31.2kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50369303(CHEMBL1204422)
Affinity DataKi:  5.00E+3nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against recombinant bovine eNOS (Endothelial nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50369301(CHEMBL1788374)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of endothelial isoform of nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50196043(3-N-(L-ArgNO2)-trans-3-amino-L-proline-NH2 ditrifl...)
Affinity DataKi:  5.76E+3nMAssay Description:Inhibition of murine macrophage iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50030279(2-Amino-5-(N'-methyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  5.90E+3nMAssay Description:Compound was tested for binding affinity against Endothelial nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061233(2-Amino-5-(N'-ethyl-guanidino)-pentanoic acid | CH...)
Affinity DataKi:  6.10E+3nMAssay Description:Compound was tested for binding affinity against recombinant inducible nitric oxide synthase (iNOS) from mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50196044(4-N-(L-ArgNO2)-Nalpha-methyl-trans-4-amino-L-proli...)
Affinity DataKi:  8.46E+3nMAssay Description:Inhibition of rat nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50061231(2-Amino-5-(N'-propyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  8.50E+3nMAssay Description:Compound was tested for binding affinity against Endothelial nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369442(CHEMBL1202118)
Affinity DataKi:  8.90E+3nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against recombinant murine Inducible nitric oxide synthase (inducible isoform)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50059651(CHEMBL96624 | omega nitro-arginine)
Affinity DataKi:  9.30E+3nMAssay Description:Compound was evaluated for the inhibition of Neuronal Nitric oxide synthase enzyme (nNOS).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50061233(2-Amino-5-(N'-ethyl-guanidino)-pentanoic acid | CH...)
Affinity DataKi:  9.50E+3nMAssay Description:Compound was tested for binding affinity against Endothelial nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50030279(2-Amino-5-(N'-methyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was tested for binding affinity against neuronal nitric oxide synthase(nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50030279(2-Amino-5-(N'-methyl-guanidino)-pentanoic acid | C...)
Affinity DataKi:  1.40E+4nMAssay Description:Compound was tested for binding affinity against recombinant inducible nitric oxide synthase (iNOS) from mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50059646(CHEMBL420996 | L-Nitroarginine-methoxy-L-phenylala...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of Neuronal Nitric oxide synthase enzyme (nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21962(3-[(4S)-4-amino-5-[(2-aminoethyl)(hydroxy)amino]pe...)
Affinity DataKi:  1.60E+4nM ΔG°:  -27.8kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50061233(2-Amino-5-(N'-ethyl-guanidino)-pentanoic acid | CH...)
Affinity DataKi:  1.60E+4nMAssay Description:Compound was tested for binding affinity against neuronal nitric oxide synthase(nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21964((2S,4R)-4-[(2S)-2-amino-N-hydroxy-5-(1-nitrocarbam...)
Affinity DataKi:  1.60E+4nM ΔG°:  -27.8kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21961((2S,4R)-4-[(2S)-2-amino-5-(1-nitrocarbamimidamido)...)
Affinity DataKi:  1.70E+4nM ΔG°:  -27.7kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50059645((2R)-2-{[(2R)-2-amino-3-phenylpropanoyl]amino}-5-{...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of Neuronal Nitric oxide synthase enzyme (nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369300(CHEMBL1202111)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of Neuronal Nitric oxide synthase enzyme (nNOS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM21960(3-[(4S)-4-amino-5-[(2-aminoethyl)amino]pentyl]-1-n...)
Affinity DataKi:  1.80E+4nM ΔG°:  -27.5kJ/molepH: 7.5 T: 2°CAssay Description:Nitric oxide formation from NOS was monitored by the hemoglobin capture assay. The assay was initiated by addition of enzyme and was monitored at 401...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50369306(CHEMBL1202112)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of inducible Nitric Oxide SynthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM22030((2S)-2-amino-N-[(1S)-3-amino-1-(aminocarbonyl)prop...)
Affinity DataKi:  2.50E+4nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against recombinant murine Inducible nitric oxide synthase (inducible isoform)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Northwestern University

LigandPNGBDBM50408718(CHEMBL2092928)
Affinity DataKi:  3.00E+4nMAssay Description:Nitric Oxide Synthase Inhibitory activity tested against recombinant bovine eNOS (Endothelial nitric oxide synthase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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