Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]-MPEP from human mGluR5More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 292nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 392nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]GR125743 from 5HT1B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.37E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5More data for this Ligand-Target Pair
Affinity DataIC50: 0.0680nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0710nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0820nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0940nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair