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Found 188 with Last Name = 'menchi' and Initial = 'g'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372593(CHEMBL410050)
Affinity DataIC50:  0.0300nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523895(CHEMBL4522121)
Affinity DataIC50:  0.0480nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372594(CHEMBL437072)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523894(CHEMBL4535400)
Affinity DataIC50:  0.0960nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523894(CHEMBL4535400)
Affinity DataIC50:  0.122nMAssay Description:Inhibition of MMP9 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  0.130nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-5 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  0.130nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372592(CHEMBL406912)
Affinity DataIC50:  0.160nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523891(CHEMBL4461597)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372596(CHEMBL270683)
Affinity DataIC50:  0.180nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50177887(CHEMBL269913 | CHEMBL556402 | c-[-Arg-Gly-Asp-Acpc...)
Affinity DataIC50:  0.260nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523890(CHEMBL4444377)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372589(CHEMBL411863)
Affinity DataIC50:  0.470nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  0.580nMAssay Description:Displacement of biotinylated ECM from human placental integrin alphavbeta3 receptor incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523891(CHEMBL4461597)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of MMP9 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372594(CHEMBL437072)
Affinity DataIC50:  0.880nMAssay Description:Displacement of [125I]echistatin from human integrin alphaVbeta5 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370689(CHEMBL392303 | ST-1646)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-5 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276748(CHEMBL460012 | [(1R,3S,9S,11S,14R)-9-(3-Guanidino-...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372591(CHEMBL406680)
Affinity DataIC50:  0.910nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523890(CHEMBL4444377)
Affinity DataIC50:  0.910nMAssay Description:Inhibition of MMP9 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372595(CHEMBL272436)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50177887(CHEMBL269913 | CHEMBL556402 | c-[-Arg-Gly-Asp-Acpc...)
Affinity DataIC50:  1.12nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-5 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372588(CHEMBL270690)
Affinity DataIC50:  1.87nMAssay Description:Displacement of [125I]echistatin from human integrin alphaVbeta5 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523897(CHEMBL4531635)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372594(CHEMBL437072)
Affinity DataIC50:  2.84nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372589(CHEMBL411863)
Affinity DataIC50:  4.40nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372588(CHEMBL270690)
Affinity DataIC50:  5.12nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor high affinity state by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372592(CHEMBL406912)
Affinity DataIC50:  5.15nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372593(CHEMBL410050)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276748(CHEMBL460012 | [(1R,3S,9S,11S,14R)-9-(3-Guanidino-...)
Affinity DataIC50:  5.64nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370689(CHEMBL392303 | ST-1646)
Affinity DataIC50:  5.64nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50092485(4-methyl-8-chloro-1,2,5,6-tetrahydro pyrido[1,2-a]...)
Affinity DataIC50:  5.80nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50276747(CHEMBL443362 | c[RGDf-(3R)-Carboxymorpholine])
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I] echistatin from alphaVbeta3 integrin isolated from human placenta after 3 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372588(CHEMBL270690)
Affinity DataIC50:  7.01nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50149341(8-Bromo-4-methyl-1,2,5,6-tetrahydro-pyrido[1,2-a]q...)
Affinity DataIC50:  8.10nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50149339(4-Methyl-8-phenylethynyl-1,2,5,6-tetrahydro-pyrido...)
Affinity DataIC50:  8.75nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523896(CHEMBL4585478)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50149329(8-Ethyl-4-methyl-1,2,5,6-tetrahydro-pyrido[1,2-a]q...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50149324(4-Methyl-8-((Z)-styryl)-1,2,5,6-tetrahydro-pyrido[...)
Affinity DataIC50:  14.2nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276746(CHEMBL452724 | c[RGDf-(3S)-Carboxymorpholine])
Affinity DataIC50:  15.1nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  18.9nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  18.9nMAssay Description:Displacement of [125I]echistatin from human integrin alpha-V-beta-3 receptor by solid phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372590(CHEMBL272661)
Affinity DataIC50:  20nMAssay Description:Inhibition of human integrin alpha-v-beta-3 receptor mediated WM115 cell adhesion to vitronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372590(CHEMBL272661)
Affinity DataIC50:  20nMAssay Description:Inhibition of human integrin alpha-V-beta-3 receptor mediated K562 cell adhesion to vitronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50092492(4,8-Dimethyl-1,2,5,6-tetrahydro-pyrido[1,2-a]quino...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276747(CHEMBL443362 | c[RGDf-(3R)-Carboxymorpholine])
Affinity DataIC50:  21nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50025356(4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type 2 in stably transfected chinese hamster ovary 1827 cells using [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523893(CHEMBL4448558)
Affinity DataIC50:  21nMAssay Description:Inhibition of MMP2 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50149335(4-Methyl-8-vinyl-1,2,5,6-tetrahydro-pyrido[1,2-a]q...)
Affinity DataIC50:  21.6nMAssay Description:Inhibitory concentration against human recombinant steroid 5-alpha-reductase type I in stably transfected chinese hamster ovary (CHO) 1827 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50523896(CHEMBL4585478)
Affinity DataIC50:  22nMAssay Description:Inhibition of MMP9 (unknown origin) pre-incubated for 5 mins before Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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