Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 31.1nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 191nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 294nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 616nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Navarra
Curated by ChEMBL
University Of Navarra
Curated by ChEMBL
Affinity DataIC50: 3.66E+3nMAssay Description:Displacement of [3H]5-HT from of SERT in rat midbrain homogenates after 5 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Navarra
Curated by ChEMBL
University Of Navarra
Curated by ChEMBL
Affinity DataIC50: 7.02E+3nMAssay Description:Displacement of [3H]5-HT from of SERT in rat midbrain homogenates after 5 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Navarra
Curated by ChEMBL
University Of Navarra
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Displacement of [3H]5-HT from of SERT in rat midbrain homogenates after 5 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Navarra
Curated by ChEMBL
University Of Navarra
Curated by ChEMBL
Affinity DataIC50: 5.78E+4nMAssay Description:Displacement of [3H]5-HT from of SERT in rat midbrain homogenates after 5 mins by scintillation countingMore data for this Ligand-Target Pair