Affinity DataKi: 0.0860nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Inhibition of recombinant human 11beta-HSD1 expressed in HEK293 cell microsomes using [3H]cortisone as substrate after 4 hrs by homogeneous immuno-ra...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair