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Found 2 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50222875'
TargetGrowth hormone secretagogue receptor type 1(Ovis aries)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50222875(6-(4-fluorophenoxy)-2-(2-methylphenyl)-3-(piperidi...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50222875(6-(4-fluorophenoxy)-2-(2-methylphenyl)-3-(piperidi...)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human recombinant GHSR1a expressed in HEK293F cells assessed as stimulation of [35S]GTP-gamma-S binding relative to ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed