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Found 44 with Last Name = 'ohmori' and Initial = 'k'
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002099(CHEMBL366965 | Dimethyl-[3-(2-methyl-6H-dibenzo[b,...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002087(4-(1-Methyl-piperidin-4-ylidene)-4,9-dihydro-1-thi...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002083(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002102(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.630nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002103(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002095(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002085(CHEMBL304185 | [11-(4-Dimethylamino-butylidene)-6,...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002086(11-(3-Pyrrolidin-1-yl-propylidene)-6,11-dihydro-di...)
Affinity DataKi:  5nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002093(CHEMBL65699 | [11-(3-Dimethylamino-propylidene)-6,...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002097(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  5.80nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002098(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040108(11-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethylsulfa...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002092(11-(3-Thiomorpholin-4-yl-propylidene)-6,11-dihydro...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002084(11-(2-Dimethylamino-ethylsulfanyl)-6,11-dihydro-di...)
Affinity DataKi:  9nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002100(11-(3-Diethylamino-propylidene)-6,11-dihydro-diben...)
Affinity DataKi:  10nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040114(CHEMBL336198 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  10nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002088(CHEMBL302005 | [11-(2-Dimethylamino-ethylidene)-6,...)
Affinity DataKi:  11nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002088(CHEMBL302005 | [11-(2-Dimethylamino-ethylidene)-6,...)
Affinity DataKi:  11nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040109(3-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  12nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002101(11-(2-Dimethylamino-ethylidene)-6,11-dihydro-diben...)
Affinity DataKi:  12nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002084(11-(2-Dimethylamino-ethylsulfanyl)-6,11-dihydro-di...)
Affinity DataKi:  14nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040112(11-[2-(4-Benzyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  14nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002089(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  15nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50175516(CHEMBL372588 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  15nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002096(ALO-4943A | CHEMBL1719 | KW-4679 | OLOPATADINE HYD...)
Affinity DataKi:  16nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040110(2-{11-[2-(4-Benzyl-piperidin-1-yl)-ethylsulfanyl]-...)
Affinity DataKi:  17nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040111(CHEMBL133080 | {11-[2-(4-Benzyl-piperidin-1-yl)-et...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002091(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040121(11-[2-(4-Phenyl-piperidin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  20nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002090(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  24nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002094(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  29nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040113(11-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethylsu...)
Affinity DataKi:  41nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040116(11-(2-Morpholin-4-yl-ethylsulfanyl)-6,11-dihydro-d...)
Affinity DataKi:  42nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040119(11-[2-(4-Phenyl-piperazin-1-yl)-ethylsulfanyl]-6,1...)
Affinity DataKi:  47nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040117(11-{2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-pi...)
Affinity DataKi:  500nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040115(CHEMBL133778 | Sodium; 11-[2-(4-benzyl-piperidin-1...)
Affinity DataKi:  740nMAssay Description:Inhibition of the specific binding of [3H]-pyrilamine to guinea pig cerebellum histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230285(CHEMBL330646)
Affinity DataIC50:  150nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230283(CHEMBL95669)
Affinity DataIC50:  520nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230288(CHEMBL321948)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230287(CHEMBL329961)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230282(CHEMBL143079)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230284(CHEMBL323555)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50230286(CHEMBL95509)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Canine Tracheal Smooth Muscle PDE 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed