Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.195nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.603nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.692nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.851nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in HEK239 cells assessed as inhibition of RAMH-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.977nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in HEK239 cells assessed as inhibition of RAMH-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.35nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.62nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair