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Found 164 with Last Name = 'perretta' and Initial = 'c'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50026614(CHEMBL575508)
Affinity DataKi:  0.0530nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027039(5''-Guanidinonaltrindole | 5''-Guanidinylnaltrindo...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214466(CHEMBL398149 | N-(3-(8-cyano-4-(cyclopropylamino)p...)
Affinity DataKi:  0.260nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  0.320nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214473(CHEMBL230354 | N-(3-(8-CYANO-4-(PHENYLAMINO)PYRAZO...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027052(CHEMBL2112473)
Affinity DataKi:  0.630nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374656(CHEMBL401544)
Affinity DataKi:  0.800nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  0.960nMAssay Description:Binding affinity towards human cloned Opioid receptor mu 1 using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50026614(CHEMBL575508)
Affinity DataKi:  1nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  1.09nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  1.10nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374653(CHEMBL271020)
Affinity DataKi:  1.30nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374662(CHEMBL256401)
Affinity DataKi:  1.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374654(CHEMBL271645)
Affinity DataKi:  1.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027052(CHEMBL2112473)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214454(CHEMBL230462 | N-(3-(8-cyano-4-(cyclobutylamino)py...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374658(CHEMBL401614)
Affinity DataKi:  2nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130561((R)-N-((S)-1-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dime...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130561((R)-N-((S)-1-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dime...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374651(CHEMBL257219)
Affinity DataKi:  2.20nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374655(CHEMBL401945)
Affinity DataKi:  2.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374657(CHEMBL257736)
Affinity DataKi:  3.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374660(CHEMBL256189)
Affinity DataKi:  3.60nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50102710(3-(4-Hydroxy-phenyl)-N-{(S)-1-[(3R,4R)-4-(3-hydrox...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027052(CHEMBL2112473)
Affinity DataKi:  3.80nMAssay Description:Binding affinity towards human cloned Opioid receptor mu 1 using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374659(CHEMBL402246)
Affinity DataKi:  4nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214465(2-(4-chlorobenzylamino)-4-(phenylamino)pyrazolo[1,...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214444(2-(p-toluidino)-4-(phenylamino)pyrazolo[1,5-a][1,3...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374661(CHEMBL402306)
Affinity DataKi:  5.20nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  5.70nMAssay Description:Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214477(4-(phenylamino)-2-(4-(pyridin-2-yl)piperazin-1-yl)...)
Affinity DataKi:  7nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50374652(CHEMBL271848)
Affinity DataKi:  7.40nMAssay Description:Inhibition of corn CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214474(CHEMBL230353 | N-(3-(8-cyano-4-(phenethylamino)pyr...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214460(2-(CYCLOHEXYLMETHYLAMINO)-4-(PHENYLAMINO)PYRAZOLO[...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50026614(CHEMBL575508)
Affinity DataKi:  8.90nMAssay Description:Binding affinity towards human cloned Opioid receptor mu 1 using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214448(2-(3,4-dimethoxyphenylamino)-4-(phenylamino)pyrazo...)
Affinity DataKi:  9nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130564(7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi:  9.80nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214464(CHEMBL230568 | N-(3-(8-methyl-4-(phenylamino)pyraz...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214450(2-(3,4-dihydroisoquinolin-2(1H)-yl)-4-(phenylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214457(2-(2,3-dihydro-1H-inden-2-ylamino)-4-(phenylamino)...)
Affinity DataKi:  12nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214453(2-(isopentylamino)-4-(phenylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027038(CHEMBL2112474)
Affinity DataKi:  13nMAssay Description:Binding affinity towards human cloned Opioid receptor mu 1 using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214468(4-(phenylamino)-2-(pyrrolidin-1-yl)pyrazolo[1,5-a]...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214446(2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine...)
Affinity DataKi:  15nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027038(CHEMBL2112474)
Affinity DataKi:  16nMAssay Description:Binding affinity towards human cloned Opioid receptor kappa 1 using [3H]U-69593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027038(CHEMBL2112474)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214443(CHEMBL230673 | N-(3-(8-bromo-4-(cyclopropylamino)p...)
Affinity DataKi:  17nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50027048(CHEMBL2112475)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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