Affinity DataKi: 4.80E+4nMAssay Description:Inhibition of mushroom tyrosinase by Lineweaver-Burke double reciprocal plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 234nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 263nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 634nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
Affinity DataIC50: 980nMAssay Description:Inhibition of mushroom tyrosine kinase assessed as oxidation of 0.25 mM L-3,4-dihydroxyphenylalanineMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 6.37E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 6.56E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 7.54E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
Affinity DataIC50: 8.33E+3nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of mushroom tyrosine kinase assessed as oxidation of 0.25 mM L-3,4-dihydroxyphenylalanineMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 9.67E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Universita Degli Studi Di Cagliari
Curated by ChEMBL
Affinity DataIC50: 6.73E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...More data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.23E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.95E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.33E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 mins by L-DOPA oxidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+6nMAssay Description:Inhibition of mushroom tyrosine kinase assessed as oxidation of 0.25 mM L-3,4-dihydroxyphenylalanineMore data for this Ligand-Target Pair