Affinity DataIC50: 0.570nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.15nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.15nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 121nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 285nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 322nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 359nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 529nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 532nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 651nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 955nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro receptor binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.75E+3nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 5.55E+3nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+4nMAssay Description:Binding affinity for Dopamine receptor D2 was assessed in vitro in rat striatal membranes using [3H]-SCH- 23390 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.67E+4nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKd: 0.127nMAssay Description:Binding affinity was determined towards serotonin uptake site in presence of [3H]-paroxetine radioligand in rat hippocampal homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKd: 0.104nMAssay Description:Binding affinity was determined towards serotonin uptake site in presence of [3H]-paroxetine radioligand in rat brain cortical homogenateMore data for this Ligand-Target Pair