Affinity DataKi: 0.800nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of human recombinant Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human recombinant Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of mouse Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition of mouse Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of mouse Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of human recombinant Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 11.8nMAssay Description:Inhibition of human recombinant Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 16.5nMAssay Description:Inhibition of mouse Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human recombinant Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 29.3nMAssay Description:Inhibition of mouse Cathepsin L assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Taigen Biotechnology
Taigen Biotechnology
Affinity DataKi: 53nM ΔG°: -41.5kJ/molepH: 7.5 T: 2°CAssay Description:The effects of compound on enzyme activity were measured by using peptide cleavage assay. Cleavage products were resolved and analyzed with a reverse...More data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Taigen Biotechnology
Taigen Biotechnology
Affinity DataKi: 58nM ΔG°: -41.3kJ/molepH: 7.5 T: 2°CAssay Description:The effects of compound on enzyme activity were measured by using peptide cleavage assay. Cleavage products were resolved and analyzed with a reverse...More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Inhibition of human recombinant Cathepsin B assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 238nMAssay Description:Inhibition of human recombinant Cathepsin B assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Inhibition of human recombinant Cathepsin B assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Taigen Biotechnology
Taigen Biotechnology
Affinity DataKi: 660nM ΔG°: -35.3kJ/molepH: 7.5 T: 2°CAssay Description:The effects of compound on enzyme activity were measured by using peptide cleavage assay. Cleavage products were resolved and analyzed with a reverse...More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 853nMAssay Description:Inhibition of human recombinant Cathepsin B assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 861nMAssay Description:Inhibition of human recombinant Cathepsin B assessed as Apparent inhibition constant using Z-FR-AMC as substrate inubated for 30 mins by fluorometric...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition constant for acetylcholinesteraseMore data for this Ligand-Target Pair