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Found 124 with Last Name = 'sydnes' and Initial = 'mo'
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375611(CHEMBL408120)
Affinity DataKi:  3.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375608(CHEMBL406220)
Affinity DataKi:  4.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375616(CHEMBL405248)
Affinity DataKi:  8nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375613(CHEMBL261577)
Affinity DataKi:  8.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375612(CHEMBL427915)
Affinity DataKi:  17.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375609(CHEMBL406283)
Affinity DataKi:  19.6nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375614(CHEMBL259235)
Affinity DataKi:  21.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375610(CHEMBL436904)
Affinity DataKi:  23.9nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375617(CHEMBL261094)
Affinity DataKi:  32.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375615(CHEMBL261583)
Affinity DataKi:  49.7nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509371(CHEMBL4521241)
Affinity DataIC50:  300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK2 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509369(CHEMBL4548361)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509369(CHEMBL4548361)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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