Compile Data Set for Download or QSAR
maximum 50k data
Found 68 with Last Name = 'tartar' and Initial = 'a'
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataKi:  4nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataKi:  170nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
TBA

Curated by ChEMBL
LigandPNGBDBM50280883((2-(2-Benzyloxycarbonylamino-2-{[(3-dimethylamino-...)
Affinity DataKi:  3.10E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTrypanothione reductase(Trypanosoma cruzi)
TBA

Curated by ChEMBL
LigandPNGBDBM50280882((3-(2-Benzyloxycarbonylamino-2-{[(3-dimethylamino-...)
Affinity DataKi:  4.30E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTrypanothione reductase(Trypanosoma cruzi)
TBA

Curated by ChEMBL
LigandPNGBDBM50280881((2-(2-Benzyloxycarbonylamino-2-{[(3-dimethylamino-...)
Affinity DataKi:  9.20E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
In DepthDetails Article
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50:  3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataIC50:  3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 microM in LLCPKI cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V2 receptor(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50:  9.5nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 microM in LLCPKI cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50:  9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataIC50:  10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataIC50:  300nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228838(CHEMBL428973)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228847(CHEMBL407100)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228846(CHEMBL265876)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50011236(CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228841(CHEMBL351282)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM15203(5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL7577...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM15203(5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL7577...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228845(CHEMBL410778)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228844(CHEMBL263188)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228842(CHEMBL437640)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  430nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  810nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  230nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  850nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152975((2S,4R)-4-Methoxy-2-(2-pyridin-2-yl-ethylthiocarba...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152976((3S,5R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  1.50E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152977((3S,5R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  1.10E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152978((3S,5R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  1.30E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152979((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  890nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152980((3S,5R)-2-([1,4'']Bipiperidinyl-1''-carbonyl)-4-me...)
Affinity DataEC50:  2.20E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152981((2S,4R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  100nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  33nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring Research

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 68 total ) | Next | Last >>
Jump to: