Compile Data Set for Download or QSAR
maximum 50k data
Found 1311 with Last Name = 'taylor' and Initial = 'e'
LigandPNGBDBM50280415((R)-2-{4-[3-(2-Amino-4-oxo-3,4,5,6,7,8-hexahydro-p...)
Affinity DataKi:  0.0000190nMAssay Description:Inhibitory activity against glycinamide ribonucleotide formyltransferase (GARFT) from L1210 murine leukemic cellsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM22590((2S)-2-[(4-{2-[(6R)-2-amino-4-oxo-1H,4H,5H,6H,7H,8...)
Affinity DataKi:  0.000120nMAssay Description:Inhibitory activity against glycinamide ribonucleotide formyltransferase (GARFT) from L1210 murine leukemic cellsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280414((R)-2-[4-(2-Amino-4-oxo-3,4,5,6,7,8-hexahydro-pyri...)
Affinity DataKi:  0.000630nMAssay Description:Inhibitory activity against glycinamide ribonucleotide formyltransferase (GARFT) from L1210 murine leukemic cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.00100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82455(BIM 23027 | BIM-23027 | N-Methylcyclo[L-Ala-L-Tyr-...)
Affinity DataKi:  0.00100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82469(BIM 23003 | BIM-23003 | EC5-21 | L-Cys(1)-L-Lys-L-...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82462(BIM 23059 | D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr...)
Affinity DataKi:  0.00800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM 23058 | BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82457((1R,4S,7S,10R,13S,16R)-4-[(R)-1-Hydroxyethyl]-7-(4...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Central Washington University

Curated by ChEMBL
LigandPNGBDBM50094929(2-(2-Methyl-piperazin-1-yl)-6-nitro-quinoline | CH...)
Affinity DataKi:  0.0810nMAssay Description:In vitro radioligand [3H]-paroxetine from rat cortical Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Central Washington University

Curated by ChEMBL
LigandPNGBDBM50063266(6-Nitro-2-piperazin-1-yl-quinoline | 6-nitroquipaz...)
Affinity DataKi:  0.163nMAssay Description:In vitro radioligand [3H]-paroxetine from rat cortical Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Central Washington University

Curated by ChEMBL
LigandPNGBDBM50063266(6-Nitro-2-piperazin-1-yl-quinoline | 6-nitroquipaz...)
Affinity DataKi:  0.163nMAssay Description:In vitro radioligand [3H]-paroxetine from rat cortical Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | MK 678 | NSC_3086456)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85052(BIM 23197 | BIM-23197)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Central Washington University

Curated by ChEMBL
LigandPNGBDBM50094930(5-Iodo-6-nitro-2-piperazin-1-yl-quinoline | CHEMBL...)
Affinity DataKi:  0.190nMAssay Description:In vitro radioligand [3H]-paroxetine from rat cortical Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  0.25nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85051(BIM-23190)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  0.880nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
Affinity DataKi:  0.930nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM85008(BIM 23066 | BIM-23066)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  1.20nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  1.22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  1.40nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  1.43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  1.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-1 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Cedars-Sinai Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-4 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82469(BIM 23003 | BIM-23003 | EC5-21 | L-Cys(1)-L-Lys-L-...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Displayed 1 to 50 (of 1311 total ) | Next | Last >>
Jump to: