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Found 5 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 2' and Ligand = 'BDBM50254239'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataEC50:  2.30nMAssay Description:Binding affinity to human SSTR2 expressed in CHO-K1 cells assessed as induction of SSTR2 internalization after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed