Affinity DataIC50: 0.160nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant human CYP1A2 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human CYP1B1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human CYP1B1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human CYP1B1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human CYP1A2 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human CYP1B1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human CYP1A1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of 2,3 dioxygenaseMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human CYP1A1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant human CYP1A1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of recombinant human CYP1A2 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of 2,3 dioxygenaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of 2,3 dioxygenaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human CYP1A1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyreso...More data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of 2,3 dioxygenaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair
TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Gyeongsang National University (Gnu)
Curated by ChEMBL
Gyeongsang National University (Gnu)
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of human leukotriene A4 hydrolaseMore data for this Ligand-Target Pair