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Found 25 with Last Name = 'thatcher' and Initial = 'ln'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218795((1R,13S,14R)-24-(cyclopropylmethyl)-20-methoxy-4,2...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109385(4-Methyl-1-(3-phenyl-propyl)-piperidine | CHEMBL35...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109384(3-Methyl-1-phenethyl-piperidine | CHEMBL144552)
Affinity DataKi:  4.20nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218793((1R,13S,14R)-20-methoxy-24-methyl-4,24-diazahexacy...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109387(3-Methyl-1-(3-phenyl-propyl)-piperidine | CHEMBL14...)
Affinity DataKi:  5.30nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109386(2-Phenethyl-1,2,3,4-tetrahydro-isoquinoline | CHEM...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109390(2-(3-Phenyl-propyl)-1,2,3,4-tetrahydro-isoquinolin...)
Affinity DataKi:  14nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218792((1R,13S,14R)-24-(cyclopropylmethyl)-19,20-dimethox...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50008585(4-Methyl-1-phenethyl-piperidine | CHEMBL343237)
Affinity DataKi:  21nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218794((1R,13S,14R)-19,20-dimethoxy-24-methyl-4,24-diazah...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218795((1R,13S,14R)-24-(cyclopropylmethyl)-20-methoxy-4,2...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DAMGO from rat recombinant mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218795((1R,13S,14R)-24-(cyclopropylmethyl)-20-methoxy-4,2...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109383(1-(3-Phenyl-propyl)-4-pyridin-2-yl-piperazine | 1-...)
Affinity DataKi:  83nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109389(1-Phenethyl-piperidine | 1-phenethylpiperidine | C...)
Affinity DataKi:  89nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]DAMGO from rat recombinant mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109391(1-(3-Phenyl-propyl)-piperidine | CHEMBL148108)
Affinity DataKi:  143nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109388(1-(2-phenylethyl)-4-(2-pyridyl)piperazine | 1-Phen...)
Affinity DataKi:  326nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218793((1R,13S,14R)-20-methoxy-24-methyl-4,24-diazahexacy...)
Affinity DataKi:  474nMAssay Description:Displacement of [3H]DAMGO from rat recombinant mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  515nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218793((1R,13S,14R)-20-methoxy-24-methyl-4,24-diazahexacy...)
Affinity DataKi:  582nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218792((1R,13S,14R)-24-(cyclopropylmethyl)-19,20-dimethox...)
Affinity DataKi:  1.44E+3nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218792((1R,13S,14R)-24-(cyclopropylmethyl)-19,20-dimethox...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]DAMGO from rat recombinant mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218794((1R,13S,14R)-19,20-dimethoxy-24-methyl-4,24-diazah...)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50218794((1R,13S,14R)-19,20-dimethoxy-24-methyl-4,24-diazah...)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [3H]DAMGO from rat recombinant mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed