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Found 519 with Last Name = 'thoresen' and Initial = 'l'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532446((1aS,5aS)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  1.45nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388463((1aS,5aS)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  1.45nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532448((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  3.80nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388466((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  3.80nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120704(2-Naphthalen-1-yl-1,3,4,5-tetrahydro-azepino[5,4,3...)
Affinity DataKi:  5nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM27685(2-{4-[(dimethylamino)methyl]phenyl}-3,10-diazatric...)
Affinity DataKi:  5nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120702(2-(4-Trifluoromethyl-phenyl)-1,3,4,5-tetrahydro-az...)
Affinity DataKi:  5nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120707(2-Thiophen-2-yl-1,3,4,5-tetrahydro-azepino[5,4,3-c...)
Affinity DataKi:  5nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120728(2-(4-Methoxy-phenyl)-1,3,4,5-tetrahydro-azepino[5,...)
Affinity DataKi:  6nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120726(2-(3-Trifluoromethyl-phenyl)-1,3,4,5-tetrahydro-az...)
Affinity DataKi:  6nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120706(2-(4-Pyrrol-1-ylmethyl-phenyl)-1,3,4,5-tetrahydro-...)
Affinity DataKi:  6nMAssay Description:In vitro inhibitory activity of the compound towards human Poly (ADP-ribose) polymerase 1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120724(2-Phenyl-1,3,4,5-tetrahydro-azepino[5,4,3-cd]indol...)
Affinity DataKi:  6nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120710(2-(3-Amino-phenyl)-1,3,4,5-tetrahydro-azepino[5,4,...)
Affinity DataKi:  7nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120721(1-Methyl-2-phenyl-1,3,4,5-tetrahydro-azepino[5,4,3...)
Affinity DataKi:  7nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120718(2-Pyridin-3-yl-1,3,4,5-tetrahydro-azepino[5,4,3-cd...)
Affinity DataKi:  7nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120723(2-(3-Dimethylaminomethyl-phenyl)-1,3,4,5-tetrahydr...)
Affinity DataKi:  8nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120731(2-(1H-Pyrrol-2-yl)-1,3,4,5-tetrahydro-azepino[5,4,...)
Affinity DataKi:  8nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120720(2-(2-Chloro-phenyl)-1,3,4,5-tetrahydro-azepino[5,4...)
Affinity DataKi:  8nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120722(2-(1H-Indol-5-yl)-1,3,4,5-tetrahydro-azepino[5,4,3...)
Affinity DataKi:  9nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120712(2-Methoxy-1,3,4,5-tetrahydro-azepino[5,4,3-cd]indo...)
Affinity DataKi:  10nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120700(6-Oxo-3,4,5,6-tetrahydro-1H-azepino[5,4,3-cd]indol...)
Affinity DataKi:  10nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120730(6-Oxo-3,4,5,6-tetrahydro-1H-azepino[5,4,3-cd]indol...)
Affinity DataKi:  11nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120709(6-Oxo-3,4,5,6-tetrahydro-1H-azepino[5,4,3-cd]indol...)
Affinity DataKi:  14nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120711(2-Benzhydryl-1,3,4,5-tetrahydro-azepino[5,4,3-cd]i...)
Affinity DataKi:  23nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120727(2-(2-Hydroxy-phenyl)-1,3,4,5-tetrahydro-azepino[5,...)
Affinity DataKi:  23nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120713(2-(4-tert-Butyl-phenyl)-1,3,4,5-tetrahydro-azepino...)
Affinity DataKi:  29nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120733(2-(2-Methylsulfanyl-phenyl)-1,3,4,5-tetrahydro-aze...)
Affinity DataKi:  32nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120701(6-Oxo-3,4,5,6-tetrahydro-1H-azepino[5,4,3-cd]indol...)
Affinity DataKi:  32nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120717(1,3,4,5-Tetrahydro-azepino[5,4,3-cd]indol-6-one | ...)
Affinity DataKi:  38nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120703(3,4-Dihydro-1H-pyrrolo[4,3,2-de]isoquinolin-5-one ...)
Affinity DataKi:  47nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120725(2-Phenyl-1,3,4,5-tetrahydro-azepino[5,4,3-cd]indol...)
Affinity DataKi:  57nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465((1aR,5aR)-2-(Tetrahydro-pyran-4-ylmethyl)-1a,2,5,5...)
Affinity DataKi:  58.7nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465((1aR,5aR)-2-(Tetrahydro-pyran-4-ylmethyl)-1a,2,5,5...)
Affinity DataKi:  58.7nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461((1aS,5aS)-2-(2,4-Difluoro-phenyl)-1a,2,5,5a-tetrah...)
Affinity DataKi:  97.6nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461((1aS,5aS)-2-(2,4-Difluoro-phenyl)-1a,2,5,5a-tetrah...)
Affinity DataKi:  97.6nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388462((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  97.7nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532445((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  97.7nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532446((1aS,5aS)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  105nMAssay Description:Table B: HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388463((1aS,5aS)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  105nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461((1aS,5aS)-2-(2,4-Difluoro-phenyl)-1a,2,5,5a-tetrah...)
Affinity DataKi:  207nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461((1aS,5aS)-2-(2,4-Difluoro-phenyl)-1a,2,5,5a-tetrah...)
Affinity DataKi:  207nMAssay Description:Table B: HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120705(2-(3,5-Bis-trifluoromethyl-phenyl)-1,3,4,5-tetrahy...)
Affinity DataKi:  230nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120714(4-(6-Oxo-3,4,5,6-tetrahydro-1H-azepino[5,4,3-cd]in...)
Affinity DataKi:  263nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120719(2-Hydroxy-1,3,4,5-tetrahydro-azepino[5,4,3-cd]indo...)
Affinity DataKi:  370nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465((1aR,5aR)-2-(Tetrahydro-pyran-4-ylmethyl)-1a,2,5,5...)
Affinity DataKi:  568nMAssay Description:Table B: HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465((1aR,5aR)-2-(Tetrahydro-pyran-4-ylmethyl)-1a,2,5,5...)
Affinity DataKi:  568nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388466((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  1.20E+3nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532448((1aR,5aR)-2-(4-Oxy-pyrazin-2-yl)-1a,2,5,5a-tetrahy...)
Affinity DataKi:  1.20E+3nMAssay Description:Table B: HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50409612(CHEMBL2112006)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120715(2-(4-Fluoro-phenyl)-3,4,5,6-tetrahydro-1H-azepino[...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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